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Open Access
Peer-reviewed
Research Article
Sulfonylpiperazine compounds prevent Plasmodium falciparum invasion of red blood cells through interference with actin-1/profilin dynamics
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Madeline G. Dans ,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Writing – original draft, Writing – review & editing
* E-mail: dans.m@wehi.edu.au (MGD); paul.gilson@burnet.edu.au (PRG)
Affiliations Burnet Institute, Melbourne, Victoria, Australia, School of Medicine and Institute for Mental and Physical Health and Clinical Translation, Deakin University, Waurn Ponds, Victoria, Australia, Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Henni Piirainen,
Roles Data curation, Formal analysis, Writing – original draft, Writing – review & editing
Affiliation Faculty of Biochemistry and Molecular Medicine, University of Oulu, Oulu, Finland
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William Nguyen,
Roles Conceptualization, Investigation, Resources, Writing – review & editing
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Sachin Khurana,
Roles Data curation, Formal analysis, Investigation, Writing – review & editing
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Somya Mehra,
Roles Data curation, Formal analysis, Writing – review & editing
Affiliation Burnet Institute, Melbourne, Victoria, Australia
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Zahra Razook,
Roles Data curation, Formal analysis, Writing – review & editing
Affiliations Burnet Institute, Melbourne, Victoria, Australia, School of Medicine and Institute for Mental and Physical Health and Clinical Translation, Deakin University, Waurn Ponds, Victoria, Australia
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Niall D. Geoghegan,
Roles Data curation, Formal analysis, Methodology
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Aurelie T. Dawson,
Roles Data curation, Methodology
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Sujaan Das,
Roles Data curation, Investigation, Methodology, Writing – review & editing
Affiliation Ludwig Maximilian University, Faculty of Veterinary Medicine, Munich, Germany
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Molly Parkyn Schneider,
Roles Data curation, Formal analysis, Writing – review & editing
Affiliation Burnet Institute, Melbourne, Victoria, Australia
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Thorey K. Jonsdottir,
Roles Data curation, Formal analysis, Writing – review & editing
Affiliations Burnet Institute, Melbourne, Victoria, Australia, Department of Microbiology and Immunology, The University of Melbourne, Parkville, Victoria, Australia
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Mikha Gabriela,
Roles Data curation, Formal analysis, Writing – review & editing
Affiliations Burnet Institute, Melbourne, Victoria, Australia, School of Medicine and Institute for Mental and Physical Health and Clinical Translation, Deakin University, Waurn Ponds, Victoria, Australia
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Maria R. Gancheva,
Roles Data curation, Methodology, Writing – review & editing
Affiliation Research Centre for Infectious Diseases, The University of Adelaide, Adelaide, Australia
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Christopher J. Tonkin,
Roles Conceptualization, Methodology, Supervision, Writing – review & editing
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Vanessa Mollard,
Roles Data curation, Formal analysis, Methodology, Writing – review & editing
Affiliation School of Biosciences, The University of Melbourne, Parkville, Victoria, Australia
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Christopher Dean Goodman,
Roles Data curation, Methodology, Writing – review & editing
Affiliation School of Biosciences, The University of Melbourne, Parkville, Victoria, Australia
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Geoffrey I. McFadden,
Roles Conceptualization, Methodology, Supervision, Writing – review & editing
Affiliation School of Biosciences, The University of Melbourne, Parkville, Victoria, Australia
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Danny W. Wilson,
Roles Conceptualization, Methodology, Supervision, Writing – review & editing
Affiliation Research Centre for Infectious Diseases, The University of Adelaide, Adelaide, Australia
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Kelly L. Rogers,
Roles Methodology, Project administration, Supervision
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Alyssa E. Barry,
Roles Methodology, Supervision, Writing – review & editing
Affiliations Burnet Institute, Melbourne, Victoria, Australia, School of Medicine and Institute for Mental and Physical Health and Clinical Translation, Deakin University, Waurn Ponds, Victoria, Australia
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Brendan S. Crabb,
Roles Funding acquisition, Supervision, Writing – review & editing
Affiliations Burnet Institute, Melbourne, Victoria, Australia, Department of Microbiology and Immunology, The University of Melbourne, Parkville, Victoria, Australia
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Tania F. de Koning-Ward,
Roles Conceptualization, Methodology, Supervision, Writing – review & editing
Affiliation School of Medicine and Institute for Mental and Physical Health and Clinical Translation, Deakin University, Waurn Ponds, Victoria, Australia
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Brad E. Sleebs,
Roles Conceptualization, Funding acquisition, Investigation, Project administration, Supervision, Writing – review & editing
Affiliation Walter and Eliza Hall Institute, Parkville, Victoria, Australia
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Inari Kursula,
Roles Conceptualization, Methodology, Supervision, Writing – review & editing
Affiliations Faculty of Biochemistry and Molecular Medicine, University of Oulu, Oulu, Finland, Department of Biomedicine, University of Bergen, Bergen, Norway
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Paul R. Gilson
Roles Conceptualization, Funding acquisition, Methodology, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: dans.m@wehi.edu.au (MGD); paul.gilson@burnet.edu.au (PRG)
Affiliations Burnet Institute, Melbourne, Victoria, Australia, Department of Microbiology and Immunology, The University of Melbourne, Parkville, Victoria, Australia
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Sulfonylpiperazine compounds prevent Plasmodium falciparum invasion of red blood cells through interference with actin-1/profilin dynamics
- Madeline G. Dans,
- Henni Piirainen,
- William Nguyen,
- Sachin Khurana,
- Somya Mehra,
- Zahra Razook,
- Niall D. Geoghegan,
- Aurelie T. Dawson,
- Sujaan Das,
- Molly Parkyn Schneider
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- Published: April 13, 2023
- https://doi.org/10.1371/journal.pbio.3002066