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Open Access
Peer-reviewed
Research Article
Structural Basis for Inhibitor-Induced Aggregation of HIV Integrase
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Kushol Gupta ,
Contributed equally to this work with: Kushol Gupta, Vesa Turkki
Affiliation Department of Biochemistry and Biophysics, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Vesa Turkki ,
Contributed equally to this work with: Kushol Gupta, Vesa Turkki
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Scott Sherrill-Mix,
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Young Hwang,
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Grant Eilers,
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Louis Taylor,
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Charlene McDanal,
Affiliation HIV DPU, Infectious Disease Therapy Area Unit GlaxoSmithKline, Research Triangle Park, North Carolina, United States of America
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Ping Wang,
Affiliation HIV DPU, Infectious Disease Therapy Area Unit GlaxoSmithKline, Research Triangle Park, North Carolina, United States of America
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David Temelkoff,
Affiliation HIV DPU, Infectious Disease Therapy Area Unit GlaxoSmithKline, Research Triangle Park, North Carolina, United States of America
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Robert T. Nolte,
Affiliation Protein Cellular and Structural Science, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Emile Velthuisen,
Affiliation HIV DPU, Infectious Disease Therapy Area Unit GlaxoSmithKline, Research Triangle Park, North Carolina, United States of America
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Jerry Jeffrey,
Affiliation HIV DPU, Infectious Disease Therapy Area Unit GlaxoSmithKline, Research Triangle Park, North Carolina, United States of America
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Gregory D. Van Duyne ,
* E-mail: vanduyne@mail.med.upenn.edu (GVD); bushman@mail.med.upenn.edu (FDB)
Affiliation Department of Biochemistry and Biophysics, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Frederic D. Bushman
* E-mail: vanduyne@mail.med.upenn.edu (GVD); bushman@mail.med.upenn.edu (FDB)
Affiliation Department of Microbiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America
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Structural Basis for Inhibitor-Induced Aggregation of HIV Integrase
- Kushol Gupta,
- Vesa Turkki,
- Scott Sherrill-Mix,
- Young Hwang,
- Grant Eilers,
- Louis Taylor,
- Charlene McDanal,
- Ping Wang,
- David Temelkoff,
- Robert T. Nolte
- Published: December 9, 2016
- https://doi.org/10.1371/journal.pbio.1002584