About the Authors

Kaleeckal G. Harikumar

Contributed equally to this work with: Kaleeckal G. Harikumar, Peishen Zhao, Brian P. Cary

Roles Formal analysis, Investigation, Writing – review & editing

Affiliation Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona, United States of America

Peishen Zhao

Contributed equally to this work with: Kaleeckal G. Harikumar, Peishen Zhao, Brian P. Cary

Roles Formal analysis, Investigation, Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Brian P. Cary

Contributed equally to this work with: Kaleeckal G. Harikumar, Peishen Zhao, Brian P. Cary

Roles Formal analysis, Investigation, Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Xiaomeng Xu

Roles Formal analysis, Investigation, Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Aditya J. Desai

Roles Formal analysis, Investigation, Writing – review & editing

Affiliation Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona, United States of America

Maoqing Dong

Roles Formal analysis, Investigation, Writing – review & editing

Affiliation Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona, United States of America

Jesse I. Mobbs

Roles Formal analysis, Investigation, Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Chirine Toufaily

Roles Writing – review & editing

Affiliation Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona, United States of America

Sebastian G. B. Furness

Roles Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, School of Biomedical Sciences, University Queensland, Queensland, Australia

Arthur Christopoulos

Roles Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Matthew J. Belousoff

Roles Formal analysis, Investigation, Writing – review & editing

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Denise Wootten

Roles Conceptualization, Formal analysis, Project administration, Supervision, Writing – original draft

denise.wootten@monash.edu (DW); patrick.sexton@monash.edu (PMS); miller@mayo.edu (LJM)

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Patrick M. Sexton

Roles Conceptualization, Formal analysis, Project administration, Supervision, Writing – original draft

denise.wootten@monash.edu (DW); patrick.sexton@monash.edu (PMS); miller@mayo.edu (LJM)

Affiliations Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia, ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia

Laurence J. Miller

Roles Conceptualization, Formal analysis, Funding acquisition, Project administration, Supervision, Writing – original draft

denise.wootten@monash.edu (DW); patrick.sexton@monash.edu (PMS); miller@mayo.edu (LJM)

Affiliation Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona, United States of America

Competing Interests

PMS and AC are co-founders and shareholders of Septerna Inc. and DACRA Tx. DW is a shareholder in Septerna Inc. and co-founder and shareholder of DACRA Tx.