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PLoS Pathogens Issue Image | Vol. 20(7) August 2024

A scheme for inhibition of AasS by C10-AMS

The AasS acyl-ACP synthetase is an exogenous fatty acid scavenger of versatility, and potentially dampens the druggable pathway of bacterial type II fatty acid synthesis. The C10-AMS compound is a newly-identified inhibitor for AasS action. This study showed complex structure of AasS hexamer liganded with C10-AMS inhibitor, of which each protomer is locked in a closed form. Huang et al

Image Credit: Youjun Feng

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A scheme for inhibition of AasS by C10-AMS

The AasS acyl-ACP synthetase is an exogenous fatty acid scavenger of versatility, and potentially dampens the druggable pathway of bacterial type II fatty acid synthesis. The C10-AMS compound is a newly-identified inhibitor for AasS action. This study showed complex structure of AasS hexamer liganded with C10-AMS inhibitor, of which each protomer is locked in a closed form. Huang et al

Image Credit: Youjun Feng

https://doi.org/10.1371/image.ppat.v20.i07.g001