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Open Access
Peer-reviewed
Research Article
Covalent Plasmodium falciparum-selective proteasome inhibitors exhibit a low propensity for generating resistance in vitro and synergize with multiple antimalarial agents
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Barbara H. Stokes,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Writing – original draft
Affiliation Department of Microbiology and Immunology, Columbia University Irving Medical Center, New York, NY, United States of America
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Euna Yoo ,
Contributed equally to this work with: Euna Yoo, James M. Murithi
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Writing – original draft
Affiliation Department of Pathology, Stanford University School of Medicine, Stanford, CA, United States of America
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James M. Murithi ,
Contributed equally to this work with: Euna Yoo, James M. Murithi
Roles Investigation
Affiliation Department of Microbiology and Immunology, Columbia University Irving Medical Center, New York, NY, United States of America
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Madeline R. Luth,
Roles Formal analysis, Investigation, Software
Affiliation Division of Host-Microbe Systems & Therapeutics, Department of Pediatrics, University of California San Diego, School of Medicine, San Diego, CA, United States of America
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Pavel Afanasyev,
Roles Formal analysis, Investigation
Affiliation MRC Laboratory of Molecular Biology, Cambridge Biomedical Campus, Cambridge, United Kingdom
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Paula C. A. da Fonseca,
Roles Resources
Affiliation MRC Laboratory of Molecular Biology, Cambridge Biomedical Campus, Cambridge, United Kingdom
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Elizabeth A. Winzeler,
Roles Resources, Software
Affiliation Division of Host-Microbe Systems & Therapeutics, Department of Pediatrics, University of California San Diego, School of Medicine, San Diego, CA, United States of America
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Caroline L. Ng ,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Validation, Writing – original draft
* E-mail: caroline.ng@unmc.edu(CLN); mbogyo@stanford.edu(MB); df2260@cumc.columbia.edu(DAF)
Current address: Department of Pathology and Microbiology, University of Nebraska Medical Center, Omaha, NE, United States of America
Affiliation Department of Microbiology and Immunology, Columbia University Irving Medical Center, New York, NY, United States of America
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Matthew Bogyo ,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Supervision, Validation, Writing – original draft
* E-mail: caroline.ng@unmc.edu(CLN); mbogyo@stanford.edu(MB); df2260@cumc.columbia.edu(DAF)
Affiliation Department of Pathology, Stanford University School of Medicine, Stanford, CA, United States of America
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David A. Fidock
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Supervision, Validation, Writing – original draft
* E-mail: caroline.ng@unmc.edu(CLN); mbogyo@stanford.edu(MB); df2260@cumc.columbia.edu(DAF)
Affiliations Department of Microbiology and Immunology, Columbia University Irving Medical Center, New York, NY, United States of America, Division of Infectious Diseases, Department of Medicine, Columbia University Irving Medical Center, New York, NY, United States of America
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Covalent Plasmodium falciparum-selective proteasome inhibitors exhibit a low propensity for generating resistance in vitro and synergize with multiple antimalarial agents
- Barbara H. Stokes,
- Euna Yoo,
- James M. Murithi,
- Madeline R. Luth,
- Pavel Afanasyev,
- Paula C. A. da Fonseca,
- Elizabeth A. Winzeler,
- Caroline L. Ng,
- Matthew Bogyo,
- David A. Fidock
- Published: June 6, 2019
- https://doi.org/10.1371/journal.ppat.1007722