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Open Access
Peer-reviewed
Research Article
Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease
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Shilpi Khare,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Steven L. Roach,
Current Address: Dart NeuroScience, San Diego, California, United States of America
Affiliation Department of Medicinal Chemistry, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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S. Whitney Barnes,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Dominic Hoepfner,
Affiliation Novartis Institutes for BioMedical Research, Novartis Campus, Basel, Switzerland
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John R. Walker,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Arnab K. Chatterjee,
Current Address: California Institute for Biomedical Research (Calibr), La Jolla, California, United States of America
Affiliation Department of Medicinal Chemistry, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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R. Jeffrey Neitz,
Affiliation Small Molecule Discovery Center and Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, United States of America
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Michelle R. Arkin,
Affiliation Small Molecule Discovery Center and Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, United States of America
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Case W. McNamara,
Current Address: California Institute for Biomedical Research (Calibr), La Jolla, California, United States of America
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Jaime Ballard,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Yin Lai,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Yue Fu,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Valentina Molteni,
Affiliation Department of Medicinal Chemistry, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Vince Yeh,
Affiliation Department of Medicinal Chemistry, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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James H. McKerrow,
Affiliation Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California, San Diego, La Jolla, California, United States of America
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Richard J. Glynne,
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Frantisek Supek
* E-mail: fsupek@gnf.org
Affiliation Department of Genetics and Neglected Diseases, Genomics Institute of the Novartis Research Foundation, San Diego, California, United States of America
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Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease
- Shilpi Khare,
- Steven L. Roach,
- S. Whitney Barnes,
- Dominic Hoepfner,
- John R. Walker,
- Arnab K. Chatterjee,
- R. Jeffrey Neitz,
- Michelle R. Arkin,
- Case W. McNamara,
- Jaime Ballard
- Published: July 17, 2015
- https://doi.org/10.1371/journal.ppat.1005058