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A mechanistic model of in vitro plasma activation to evaluate therapeutic kallikrein-kinin system inhibitors

Fig 7

Inhibition of BK generation via different KKS inhibitors.

a) Simulated data showing the proportion of CSL312-FXII complex to total FXII in plasma equilibrated with different concentrations of CSL312, b) normalised BK concentrations generated by DXS-mediated activation of healthy pooled plasma titrated with various KKS inhibitors, comparison of in vitro data with model output. Experimental data was adapted from Cao et al. [8].

Fig 7

doi: https://doi.org/10.1371/journal.pcbi.1012552.g007