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Open Access
Peer-reviewed
Research Article
Predicting kinase inhibitors using bioactivity matrix derived informer sets
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Huikun Zhang ,
Contributed equally to this work with: Huikun Zhang, Spencer S. Ericksen, Ching-pei Lee
Roles Formal analysis, Investigation, Methodology, Software, Writing – original draft
Affiliation Department of Statistics, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Spencer S. Ericksen ,
Contributed equally to this work with: Huikun Zhang, Spencer S. Ericksen, Ching-pei Lee
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Software, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Small Molecule Screening Facility, Drug Development Core, UW-Carbone Cancer Center, School of Medicine and Public Health, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Ching-pei Lee ,
Contributed equally to this work with: Huikun Zhang, Spencer S. Ericksen, Ching-pei Lee
Roles Formal analysis, Investigation, Methodology, Software, Writing – original draft
Affiliation Department of Mathematics and Institute for Mathematical Science, National University of Singapore, Singapore
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Gene E. Ananiev,
Roles Data curation, Investigation
Affiliation Small Molecule Screening Facility, Drug Development Core, UW-Carbone Cancer Center, School of Medicine and Public Health, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Nathan Wlodarchak,
Roles Data curation, Investigation, Resources, Writing – review & editing
Affiliation Department of Medicine, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Peng Yu,
Roles Formal analysis, Investigation
Affiliation Department of Statistics, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Julie C. Mitchell,
Roles Conceptualization, Funding acquisition, Writing – review & editing
Affiliation Biosciences Division, Oak Ridge National Laboratory, Oak Ridge, Tennesse, United States of America
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Anthony Gitter,
Roles Conceptualization, Funding acquisition, Software, Supervision, Validation, Writing – review & editing
Affiliations Department of Biostatistics and Medical Informatics, University of Wisconsin-Madison, Madison, Wisconsin, United States of America, Morgridge Institute for Research, Madison, Wisconsin, United States of America
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Stephen J. Wright,
Roles Conceptualization, Formal analysis, Funding acquisition, Methodology, Project administration, Software, Supervision, Writing – review & editing
Affiliation Department of Computer Sciences, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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F. Michael Hoffmann,
Roles Conceptualization, Funding acquisition, Project administration, Supervision, Writing – original draft, Writing – review & editing
Affiliations Small Molecule Screening Facility, Drug Development Core, UW-Carbone Cancer Center, School of Medicine and Public Health, University of Wisconsin-Madison, Madison, Wisconsin, United States of America, Department of Oncology, McArdle Laboratory for Cancer Research, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Scott A. Wildman,
Roles Conceptualization, Investigation, Methodology, Project administration, Supervision, Writing – original draft, Writing – review & editing
Affiliation Small Molecule Screening Facility, Drug Development Core, UW-Carbone Cancer Center, School of Medicine and Public Health, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Michael A. Newton
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Software, Supervision, Visualization, Writing – original draft, Writing – review & editing
* E-mail: newton@stat.wisc.edu
Affiliations Department of Statistics, University of Wisconsin-Madison, Madison, Wisconsin, United States of America, Department of Biostatistics and Medical Informatics, University of Wisconsin-Madison, Madison, Wisconsin, United States of America
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Predicting kinase inhibitors using bioactivity matrix derived informer sets
- Huikun Zhang,
- Spencer S. Ericksen,
- Ching-pei Lee,
- Gene E. Ananiev,
- Nathan Wlodarchak,
- Peng Yu,
- Julie C. Mitchell,
- Anthony Gitter,
- Stephen J. Wright,
- F. Michael Hoffmann
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- Published: August 5, 2019
- https://doi.org/10.1371/journal.pcbi.1006813