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Partial agonists

In Vitro and In Vivo Characterization of the Alkaloid Nuciferine

Martilias S. Farrell, John D. McCorvy, Xi-Ping Huang, Daniel J. Urban, Kate L. White, Patrick M. Giguere, Allison K. Doak, Alison I. Bernstein, Kristen A. Stout, Su Mi Park, Ramona M. Rodriguiz, Bradley W. Gray, William S. Hyatt, Andrew P. Norwood, Kevin A. Webster, Brenda M. Gannon, Gary W. Miller, Joseph H. Porter, Brian K. Shoichet, William E. Fantegrossi, William C. Wetsel, Bryan L. Roth

published 10 Mar 2016

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Nicotinic Activity of Arecoline, the Psychoactive Element of "Betel Nuts", Suggests a Basis for Habitual Use and Anti-Inflammatory Activity

Roger L. Papke, Nicole A. Horenstein, Clare Stokes

published 21 Oct 2015

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Similarities and Distinctions in Actions of Surface-Directed and Classic Androgen Receptor Antagonists

Ji Ho Suh, Arundhati Chattopadhyay, Douglas H. Sieglaff, Cheryl Storer Samaniego, Marc B. Cox, Paul Webb

published 02 Sep 2015

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Pharmacological Profile of Nociceptin/Orphanin FQ Receptors Interacting with G-Proteins and β-Arrestins 2

D. Malfacini, C. Ambrosio, M. C. Gro’, M. Sbraccia, C. Trapella, R. Guerrini, M. Bonora, P. Pinton, T. Costa, G. Calo’

published 06 Aug 2015

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Differential Effects of D-Cycloserine and ACBC at NMDA Receptors in the Rat Entorhinal Cortex Are Related to Efficacy at the Co-Agonist Binding Site

Alex M. Lench, Emma Robson, Roland S. G. Jones

published 20 Jul 2015

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Unique Effects of Acute Aripiprazole Treatment on the Dopamine D2 Receptor Downstream cAMP-PKA and Akt-GSK3β Signalling Pathways in Rats

Bo Pan, Jiezhong Chen, Jiamei Lian, Xu-Feng Huang, Chao Deng

published 10 Jul 2015

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Phosphorylation of PPARγ Affects the Collective Motions of the PPARγ-RXRα-DNA Complex

Justin A. Lemkul, Stephanie N. Lewis, Josep Bassaganya-Riera, David R. Bevan

published 08 May 2015

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An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor β (RARβ, NR1B2) Selective Agonist

Eswarkumar Nadendla, Catherine Teyssier, Vanessa Delfosse, Valérie Vivat, Gunasekaran Krishnasamy, Hinrich Gronemeyer, William Bourguet, Pierre Germain

published 01 May 2015

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Antipsychotic-Like Effect of the Muscarinic Acetylcholine Receptor Agonist BuTAC in Non-Human Primates

Maibritt B. Andersen, Carrie Hughes Croy, Ditte Dencker, Thomas Werge, Frank P. Bymaster, Christian C. Felder, Anders Fink-Jensen

published 16 Apr 2015

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The Extracellular Loop 2 (ECL2) of the Human Histamine H₄ Receptor Substantially Contributes to Ligand Binding and Constitutive Activity

David Wifling, Günther Bernhardt, Stefan Dove, Armin Buschauer

published 28 Jan 2015

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Ligand-Dependent Opening of the Multiple AMPA Receptor Conductance States: A Concerted Model

Ranjita Dutta-Roy, Christian Rosenmund, Stuart J. Edelstein, Nicolas Le Novère

published 28 Jan 2015

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Active-State Model of a Dopamine D₂ Receptor - Gα_i Complex Stabilized by Aripiprazole-Type Partial Agonists

Ralf C. Kling, Nuska Tschammer, Harald Lanig, Timothy Clark, Peter Gmeiner

published 16 Jun 2014

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Extending the Applicability of the Dose Addition Model to the Assessment of Chemical Mixtures of Partial Agonists by Using a Novel Toxic Unit Extrapolation Method

Martin Scholze, Elisabete Silva, Andreas Kortenkamp

published 12 Feb 2014

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