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Open Access
Peer-reviewed
Research Article
Inhibition of prenylated KRAS in a lipid environment
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Johanna M. Jansen ,
* E-mail: johanna.jansen@novartis.com
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Charles Wartchow,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Wolfgang Jahnke,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Susan Fong,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Tiffany Tsang,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Keith Pfister,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Tatiana Zavorotinskaya,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Dirksen Bussiere,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Jan Marie Cheng,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Kenneth Crawford,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Yumin Dai,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Jeffrey Dove,
Current address: Edison Pharmaceuticals, Mountain View, California, United States of America
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Eric Fang,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Yun Feng,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Cambridge, Massachusetts, United States of America
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Jean-Michel Florent,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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John Fuller,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Alvar D. Gossert,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Mohammad Hekmat-Nejad,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Chrystèle Henry,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Julia Klopp,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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William P. Lenahan †,
† Deceased.
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Andreas Lingel,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Sylvia Ma,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Arndt Meyer,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Yuji Mishina,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Cambridge, Massachusetts, United States of America
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Jamie Narberes,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Gwynn Pardee,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Savithri Ramurthy,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Sebastien Rieffel,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Darrin Stuart,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Cambridge, Massachusetts, United States of America
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Sharadha Subramanian,
Affiliation Department of Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Laura Tandeske,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Stephania Widger,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Armin Widmer,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Aurelie Winterhalter,
Affiliation Center for Proteomic Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland
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Isabel Zaror,
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
⨯ - [ ... ],
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Stephen Hardy
Affiliation Department of Oncology, Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Inhibition of prenylated KRAS in a lipid environment
- Johanna M. Jansen,
- Charles Wartchow,
- Wolfgang Jahnke,
- Susan Fong,
- Tiffany Tsang,
- Keith Pfister,
- Tatiana Zavorotinskaya,
- Dirksen Bussiere,
- Jan Marie Cheng,
- Kenneth Crawford
- Published: April 6, 2017
- https://doi.org/10.1371/journal.pone.0174706