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Open Access
Peer-reviewed
Research Article
Kinome analysis of Madurella mycetomatis identified kinases in the cell wall integrity pathway as novel potential therapeutic drug targets in eumycetoma caused by Madurella mycetomatis
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Mickey Konings,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Visualization, Writing – original draft
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Nikolaos Strepis,
Roles Formal analysis, Investigation, Methodology, Visualization, Writing – review & editing
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Ri-Ichiroh Manabe,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Laboratory for Comprehensive Genomic Analysis, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan
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Akira Hasegawa,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Laboratory for Large-Scale Biomedical Data Technology, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan
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Somdatta Chaudhari,
Roles Formal analysis, Investigation, Methodology, Resources, Software, Visualization, Writing – review & editing
Affiliation Department of Pharmaceutical Chemistry, Progressive Education society’s Modern College of Pharmacy, Pune, Maharashtra, India
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Saskia du Pré,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Marij Schippers,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Michihira Tagami,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Laboratory for Comprehensive Genomic Analysis, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan
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Jingyi Ma,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Yasushi Okazaki,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Laboratory for Comprehensive Genomic Analysis, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan
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Matthew Todd,
Roles Conceptualization, Investigation, Methodology, Visualization, Writing – review & editing
Affiliation School of Pharmacy and Structural Genomics Consortium, University College London, London, United Kingdom
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Bernhard Biersack,
Roles Resources, Visualization, Writing – review & editing
Affiliation Organic Chemistry Laboratory, University Bayreuth, Bayreuth, Germany
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Vijay Masand,
Roles Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Department of Chemistry, Vidya Bharati Mahavidyalaya, Amravati, Maharashtra, India
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Annelies Verbon,
Roles Supervision, Writing – review & editing
Affiliations Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands, Department of Internal Medicine, UMC Utrecht, Utrecht, The Netherlands
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Takeya Kasukawa,
Roles Conceptualization, Supervision, Writing – review & editing
Affiliation Laboratory for Large-Scale Biomedical Data Technology, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan
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Imad Abugessaisa ,
Roles Conceptualization, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Software, Visualization, Writing – original draft, Writing – review & editing
* E-mail: w.vandesande@erasmusmc.nl (WWJS); abugessaisa.prime@osaka-u.ac.jp (IA)
Affiliations Laboratory for Large-Scale Biomedical Data Technology, RIKEN Center for Integrative Medical Sciences, Yokohama, Kanagawa, Japan, Premium Research Institute for Human Metaverse Medicine (WPI-PRIMe), The University of Osaka, Suita, Osaka, Japan, Graduate School of Medicine and Faculty of Medicine, The University of Osaka, Suita, Osaka, Japan
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Wendy W. J. van de Sande
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Supervision, Visualization, Writing – original draft, Writing – review & editing
* E-mail: w.vandesande@erasmusmc.nl (WWJS); abugessaisa.prime@osaka-u.ac.jp (IA)
Affiliation Department of Medical Microbiology and Infectious Diseases Rotterdam, Erasmus Medical Center, University Medical Centre, Rotterdam, The Netherlands
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Kinome analysis of Madurella mycetomatis identified kinases in the cell wall integrity pathway as novel potential therapeutic drug targets in eumycetoma caused by Madurella mycetomatis
- Mickey Konings,
- Nikolaos Strepis,
- Ri-Ichiroh Manabe,
- Akira Hasegawa,
- Somdatta Chaudhari,
- Saskia du Pré,
- Marij Schippers,
- Michihira Tagami,
- Jingyi Ma,
- Yasushi Okazaki
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- Published: September 4, 2025
- https://doi.org/10.1371/journal.pntd.0013482