-
Loading metrics
Open Access
Peer-reviewed
Research Article
Discovery of ABBV-4083, a novel analog of Tylosin A that has potent anti-Wolbachia and anti-filarial activity
-
Thomas W. von Geldern ,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Writing – original draft, Writing – review & editing
* E-mail: thomas.vongeldern@abbvie.com, tvongeldern@earthlink.net
Affiliations Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America, Franciscan Institute for World Health, Franciscan University, Steubenville, Ohio, United States of America
⨯ -
Howard E. Morton,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Writing – review & editing
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Rick F. Clark,
Roles Conceptualization, Investigation, Writing – review & editing
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Brian S. Brown,
Roles Conceptualization, Investigation, Writing – review & editing
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Kelly L. Johnston,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Liverpool, United Kingdom
⨯ -
Louise Ford,
Roles Data curation, Investigation, Methodology, Writing – review & editing
Affiliation Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Liverpool, United Kingdom
⨯ -
Sabine Specht,
Roles Data curation, Formal analysis, Investigation, Methodology, Visualization
Current address: Filariasis Program, Drugs for Neglected Diseases Initiative, Geneva, Switzerland.
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Robert A. Carr,
Roles Data curation, Formal analysis, Investigation
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Deanne F. Stolarik,
Roles Investigation, Methodology
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Junli Ma,
Roles Investigation, Methodology
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Matthew J. Rieser,
Roles Investigation, Methodology
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ -
Dominique Struever,
Roles Investigation, Methodology
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Stefan J. Frohberger,
Roles Investigation, Methodology
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Marianne Koschel,
Roles Investigation, Methodology
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Alexandra Ehrens,
Roles Investigation, Methodology
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Joseph D. Turner,
Roles Conceptualization, Formal analysis, Writing – review & editing
Affiliation Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Liverpool, United Kingdom
⨯ -
Marc P. Hübner,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Supervision, Visualization, Writing – review & editing
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Achim Hoerauf,
Roles Conceptualization, Funding acquisition, Investigation, Project administration, Resources, Supervision
Affiliation Institute for Medical Microbiology, Immunology and Parasitology, University Hospital, Bonn, Germany
⨯ -
Mark J. Taylor,
Roles Conceptualization, Funding acquisition, Project administration, Resources, Supervision
Affiliation Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Liverpool, United Kingdom
⨯ -
Stephen A. Ward,
Roles Conceptualization, Funding acquisition, Project administration, Resources, Supervision
Affiliation Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Liverpool, United Kingdom
⨯ -
Kennan Marsh,
Roles Data curation, Formal analysis, Investigation, Methodology, Supervision, Writing – review & editing
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ - [ ... ],
-
Dale J. Kempf
Roles Conceptualization, Funding acquisition, Investigation, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing
Affiliation Global Pharmaceutical Research and Development, AbbVie, North Chicago, Illinois, United States of America
⨯ - [ view all ]
- [ view less ]
Discovery of ABBV-4083, a novel analog of Tylosin A that has potent anti-Wolbachia and anti-filarial activity
- Thomas W. von Geldern,
- Howard E. Morton,
- Rick F. Clark,
- Brian S. Brown,
- Kelly L. Johnston,
- Louise Ford,
- Sabine Specht,
- Robert A. Carr,
- Deanne F. Stolarik,
- Junli Ma
-
- Published: February 28, 2019
- https://doi.org/10.1371/journal.pntd.0007159