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Open Access
Peer-reviewed
Research Article
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents
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Dana M. Klug,
Roles Conceptualization, Formal analysis, Investigation, Writing – original draft, Writing – review & editing
Affiliation Northeastern University Department of Chemistry & Chemical Biology, Boston, MA, United States of America
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Rosario Diaz-Gonzalez,
Roles Conceptualization, Investigation, Methodology, Supervision, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Guiomar Pérez-Moreno,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Gloria Ceballos-Pérez,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Raquel García-Hernández,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Veronica Gomez-Pérez,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Luis Miguel Ruiz-Pérez,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Domingo I. Rojas-Barros,
Roles Investigation, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Francisco Gamarro,
Roles Funding acquisition, Investigation, Project administration, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Dolores González-Pacanowska,
Roles Funding acquisition, Investigation, Project administration, Validation
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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María S. Martínez-Martínez,
Roles Investigation, Validation
Affiliation Tres Cantos Medicines Development Campus, DDW and CIB, GlaxoSmithKline, Tres Cantos, Spain
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Pilar Manzano,
Roles Conceptualization, Investigation, Supervision, Validation
Affiliation Tres Cantos Medicines Development Campus, DDW and CIB, GlaxoSmithKline, Tres Cantos, Spain
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Lori Ferrins,
Roles Project administration, Writing – review & editing
Affiliation Northeastern University Department of Chemistry & Chemical Biology, Boston, MA, United States of America
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Conor R. Caffrey,
Roles Investigation, Supervision, Validation
Affiliation Center for Discovery and Innovation in Parasitic Diseases, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California, San Diego, La Jolla, CA, United States of America
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Miguel Navarro,
Roles Conceptualization, Funding acquisition, Project administration, Supervision
Affiliation Instituto de Parasitología y Biomedicina “López-Neyra” Consejo Superior de Investigaciones Cientificas (CSIC), Granada, Spain
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Michael P. Pollastri
Roles Conceptualization, Funding acquisition, Project administration, Supervision, Writing – review & editing
* E-mail: m.pollastri@northeastern.edu
Affiliation Northeastern University Department of Chemistry & Chemical Biology, Boston, MA, United States of America
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Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents
- Dana M. Klug,
- Rosario Diaz-Gonzalez,
- Guiomar Pérez-Moreno,
- Gloria Ceballos-Pérez,
- Raquel García-Hernández,
- Veronica Gomez-Pérez,
- Luis Miguel Ruiz-Pérez,
- Domingo I. Rojas-Barros,
- Francisco Gamarro,
- Dolores González-Pacanowska
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- Published: February 8, 2019
- https://doi.org/10.1371/journal.pntd.0007129