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Open Access
Peer-reviewed
Research Article
Discovery of novel, orally bioavailable, antileishmanial compounds using phenotypic screening
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Diana Ortiz ,
Roles Data curation, Formal analysis, Investigation, Methodology, Supervision, Writing – original draft, Writing – review & editing
¶‡ These authors are designated as joint first authors
Affiliation Department of Molecular Microbiology & Immunology, Oregon Health & Science University, Portland, Oregon, United States of America
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W. Armand Guiguemde ,
Roles Data curation, Formal analysis, Investigation, Methodology, Supervision
¶‡ These authors are designated as joint first authors
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Jared T. Hammill,
Roles Data curation, Formal analysis, Methodology, Writing – original draft, Writing – review & editing
Current address: Department of Pharmaceutical Sciences, University of Kentucky, Lexington, KY United States of America
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Angela K. Carrillo,
Roles Data curation, Formal analysis, Writing – original draft
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Yizhe Chen,
Roles Data curation, Formal analysis, Methodology, Resources
Current address: Department of Pharmaceutical Sciences, University of Kentucky, Lexington, KY United States of America
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Michele Connelly,
Roles Data curation, Formal analysis, Investigation, Resources
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Kayla Stalheim,
Roles Formal analysis, Investigation
Affiliation Department of Molecular Microbiology & Immunology, Oregon Health & Science University, Portland, Oregon, United States of America
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Carolyn Elya,
Roles Data curation, Formal analysis, Investigation, Methodology
Affiliation Department of Molecular Microbiology & Immunology, Oregon Health & Science University, Portland, Oregon, United States of America
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Alex Johnson,
Roles Formal analysis, Investigation
Affiliation Department of Molecular Microbiology & Immunology, Oregon Health & Science University, Portland, Oregon, United States of America
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Jaeki Min,
Roles Data curation, Formal analysis, Investigation, Resources, Supervision
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Anang Shelat,
Roles Data curation, Formal analysis, Investigation
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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David C. Smithson,
Roles Data curation, Formal analysis, Investigation, Methodology, Supervision
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Lei Yang,
Roles Formal analysis, Investigation, Methodology
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Fangyi Zhu,
Roles Formal analysis, Investigation, Methodology, Resources
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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R. Kiplin Guy ,
Roles Conceptualization, Formal analysis, Funding acquisition, Methodology, Project administration, Supervision, Writing – review & editing
* E-mail: landfear@ohsu.edu (SML); kip.guy@uky.edu (RKG)
Current address: Department of Pharmaceutical Sciences, University of Kentucky, Lexington, KY United States of America
Affiliation Department of Chemical Biology and Theraputics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United States of America
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Scott M. Landfear
Roles Conceptualization, Formal analysis, Funding acquisition, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: landfear@ohsu.edu (SML); kip.guy@uky.edu (RKG)
Affiliation Department of Molecular Microbiology & Immunology, Oregon Health & Science University, Portland, Oregon, United States of America
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Discovery of novel, orally bioavailable, antileishmanial compounds using phenotypic screening
- Diana Ortiz,
- W. Armand Guiguemde,
- Jared T. Hammill,
- Angela K. Carrillo,
- Yizhe Chen,
- Michele Connelly,
- Kayla Stalheim,
- Carolyn Elya,
- Alex Johnson,
- Jaeki Min
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- Published: December 29, 2017
- https://doi.org/10.1371/journal.pntd.0006157