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Open Access
Peer-reviewed
Research Article
Design and synthesis of novel anti-urease imidazothiazole derivatives with promising antibacterial activity against Helicobacter pylori
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Afnan I. Shahin,
Roles Investigation, Methodology, Writing – original draft, Writing – review & editing
Affiliation Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates
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Sumera Zaib ,
Roles Conceptualization, Data curation, Supervision, Writing – original draft, Writing – review & editing
* E-mail: drmelgamal2002@gmail.com, malgamal@sharjah.ac.ae, drmelgamal@mans.edu.eg (MIEG); gkhoder@sharjah.ac.ae (GK); sumera.biochem@gmail.com, sumera.zaib@ucp.edu.pk (SZ)
Affiliation Faculty of Science and Technology, Department of Basic and Applied Chemistry, University of Central Punjab, Lahore, Pakistan
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Seyed-Omar Zaraei,
Roles Data curation, Investigation, Writing – original draft, Writing – review & editing
Affiliation Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates
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Reena A. Kedia,
Roles Data curation, Investigation, Methodology
Affiliation Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates
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Hanan S. Anbar,
Roles Conceptualization, Investigation, Methodology, Writing – original draft, Writing – review & editing
Affiliation Department of Clinical Pharmacy and Pharmacotherapeutics, Dubai Pharmacy College for Girls, Dubai, United Arab Emirates
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Muhammad Tayyab Younas,
Roles Data curation, Investigation, Methodology
Affiliation Faculty of Science and Technology, Department of Basic and Applied Chemistry, University of Central Punjab, Lahore, Pakistan
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Taleb H. Al-Tel,
Roles Conceptualization, Supervision, Writing – original draft, Writing – review & editing
Affiliations Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates, Department of Medicinal Chemistry, College of Pharmacy, University of Sharjah, Sharjah, United Arab Emirates
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Ghalia Khoder ,
Roles Conceptualization, Data curation, Funding acquisition, Project administration, Writing – original draft, Writing – review & editing
* E-mail: drmelgamal2002@gmail.com, malgamal@sharjah.ac.ae, drmelgamal@mans.edu.eg (MIEG); gkhoder@sharjah.ac.ae (GK); sumera.biochem@gmail.com, sumera.zaib@ucp.edu.pk (SZ)
Affiliations Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates, Department of Pharmaceutics and Pharmaceutical Technology, College of Pharmacy, University of Sharjah, Sharjah, United Arab Emirates
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Mohammed I. El-Gamal
Roles Conceptualization, Funding acquisition, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: drmelgamal2002@gmail.com, malgamal@sharjah.ac.ae, drmelgamal@mans.edu.eg (MIEG); gkhoder@sharjah.ac.ae (GK); sumera.biochem@gmail.com, sumera.zaib@ucp.edu.pk (SZ)
Affiliations Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates, Department of Medicinal Chemistry, College of Pharmacy, University of Sharjah, Sharjah, United Arab Emirates, Faculty of Pharmacy, Department of Medicinal Chemistry, Mansoura University, Mansoura, Egypt
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Design and synthesis of novel anti-urease imidazothiazole derivatives with promising antibacterial activity against Helicobacter pylori
- Afnan I. Shahin,
- Sumera Zaib,
- Seyed-Omar Zaraei,
- Reena A. Kedia,
- Hanan S. Anbar,
- Muhammad Tayyab Younas,
- Taleb H. Al-Tel,
- Ghalia Khoder,
- Mohammed I. El-Gamal
- Published: June 2, 2023
- https://doi.org/10.1371/journal.pone.0286684