Identification of a novel CDK9 inhibitor targeting the intramolecular hidden cavity of CDK9 induced by Tat binding

• Kaori Asamitsu ,

  Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Software, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing

  * E-mail: asamitsu@med.nagoya-cu.ac.jp (KA); t-hirokawa@md.tsukuba.ac.jp (TH)

  Affiliation Department of Neurocognitive Science, Institute of Brain Science, Graduate School of Medical Sciences, Nagoya City University, Nagoya, Aichi, Japan

  https://orcid.org/0000-0001-5333-8011

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• Takatsugu Hirokawa ,

  Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Software, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing

  * E-mail: asamitsu@med.nagoya-cu.ac.jp (KA); t-hirokawa@md.tsukuba.ac.jp (TH)

  Affiliations Division of Biomedical Science, Faculty of Medicine, University of Tsukuba, Tsukuba, Ibaragi, Japan, Transborder Medical Research Center, University of Tsukuba, Tsukuba, Ibaragi, Japan

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• Takashi Okamoto

  Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Software, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing

  Affiliation Department of Neurocognitive Science, Institute of Brain Science, Graduate School of Medical Sciences, Nagoya City University, Nagoya, Aichi, Japan

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