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Open Access
Peer-reviewed
Research Article
Chirality and asymmetry increase the potency of candidate ADRM1/RPN13 inhibitors
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Ravi K. Anchoori,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliations Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America, Department of Oncology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Logan George,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Visualization, Writing – original draft
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Ssu-Hsueh Tseng,
Roles Data curation, Formal analysis, Investigation, Methodology, Visualization
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Brandon Lam,
Roles Data curation, Formal analysis, Investigation, Methodology, Resources
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Srinidhi Polkampally,
Roles Investigation, Methodology, Validation, Visualization
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Anjali D. Amiano,
Roles Investigation, Methodology, Validation, Visualization
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Palmer Foran,
Roles Investigation, Methodology, Visualization
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Hannah Tsingine,
Roles Conceptualization, Data curation, Investigation, Writing – review & editing
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Harideep Samanapally,
Roles Investigation, Methodology, Visualization
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Fernanda Carrizo Velasquez,
Roles Data curation, Formal analysis, Investigation, Methodology, Visualization
Affiliations Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America, Department of Anesthesiology and Critical Care Medicine, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Samarjit Das,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliations Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America, Department of Anesthesiology and Critical Care Medicine, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Deyin Xing,
Roles Methodology, Resources, Supervision, Writing – review & editing
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Ahmad Bin Salam,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Resources, Software
Affiliation Department of Biology and Center for Cancer Research, Tuskegee University, Tuskegee, Alabama, United States of America
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Balasubramanyam Karanam,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Software, Writing – original draft, Writing – review & editing
Affiliation Department of Biology and Center for Cancer Research, Tuskegee University, Tuskegee, Alabama, United States of America
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Chien-Fu Hung,
Roles Conceptualization, Funding acquisition, Methodology, Resources, Supervision, Writing – original draft, Writing – review & editing
Affiliation Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Richard B. S. Roden
Roles Conceptualization, Data curation, Funding acquisition, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing
* E-mail: roden@jhmi.edu
Affiliations Department of Pathology, The Johns Hopkins University, Baltimore, Maryland, United States of America, Department of Oncology, The Johns Hopkins University, Baltimore, Maryland, United States of America, Department of Gynecology & Obstetrics, The Johns Hopkins University, Baltimore, Maryland, United States of America
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Chirality and asymmetry increase the potency of candidate ADRM1/RPN13 inhibitors
- Ravi K. Anchoori,
- Logan George,
- Ssu-Hsueh Tseng,
- Brandon Lam,
- Srinidhi Polkampally,
- Anjali D. Amiano,
- Palmer Foran,
- Hannah Tsingine,
- Harideep Samanapally,
- Fernanda Carrizo Velasquez
- Published: September 10, 2021
- https://doi.org/10.1371/journal.pone.0256937