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Open Access
Peer-reviewed
Research Article
Development of an orally-administrable tumor vasculature-targeting therapeutic using annexin A1-binding D-peptides
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Motohiro Nonaka,
Roles Data curation, Investigation, Methodology, Software, Validation, Visualization, Writing – original draft
Affiliations Laboratory for Drug Discovery, National Institute of Advanced Industrial Science and Technology, Tsukuba, Ibaraki, Japan, Department of Biological Chemistry, Human Health Sciences, Graduate School of Medicine, Kyoto University, Kyoto, Japan
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Hideaki Mabashi-Asazuma,
Roles Data curation, Methodology, Resources, Validation
Affiliation Department of Molecular Biology, University of Wyoming, Laramie, WY, United States of America
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Donald L. Jarvis,
Roles Funding acquisition, Investigation, Methodology, Software, Validation
Affiliation Department of Molecular Biology, University of Wyoming, Laramie, WY, United States of America
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Kazuhiko Yamasaki,
Roles Investigation, Methodology, Software, Validation
Affiliation Biomedical Research Institute, National Institute of Advanced Industrial Science and Technology, Tsukuba, Ibaraki, Japan
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Tomoya O. Akama,
Roles Data curation, Investigation, Methodology, Validation
Affiliation Department of Pharmacology, Kansai Medical University, Hirakata, Osaka, Japan
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Masato Nagaoka,
Roles Data curation, Formal analysis, Investigation, Methodology, Resources, Software, Supervision, Validation
Affiliation Yakult Central Institute, Kunitachi, Tokyo, Japan
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Toshio Sasai,
Roles Data curation, Investigation, Methodology, Software, Validation
Affiliation Yakult Central Institute, Kunitachi, Tokyo, Japan
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Itsuko Kimura-Takagi,
Roles Data curation, Investigation, Methodology
Affiliation Yakult Central Institute, Kunitachi, Tokyo, Japan
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Yoichi Suwa,
Roles Data curation, Methodology, Resources, Software, Validation
Affiliation Yakult Central Institute, Kunitachi, Tokyo, Japan
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Takashi Yaegashi,
Roles Investigation, Methodology, Resources, Validation
Affiliation Yakult Central Institute, Kunitachi, Tokyo, Japan
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Chun-Teng Huang,
Roles Investigation, Methodology, Resources
Affiliation Cancer Center, Sanford-Burnham-Prebys Medical Discovery Institute, La Jolla, CA, United States of America
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Chizuko Nishizawa-Harada,
Roles Data curation, Investigation, Methodology, Validation
Affiliation Laboratory for Drug Discovery, National Institute of Advanced Industrial Science and Technology, Tsukuba, Ibaraki, Japan
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Michiko N. Fukuda
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Supervision, Validation, Writing – original draft, Writing – review & editing
* E-mail: michiko@sbpdiscovery.org
Affiliations Laboratory for Drug Discovery, National Institute of Advanced Industrial Science and Technology, Tsukuba, Ibaraki, Japan, Cancer Center, Sanford-Burnham-Prebys Medical Discovery Institute, La Jolla, CA, United States of America
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Development of an orally-administrable tumor vasculature-targeting therapeutic using annexin A1-binding D-peptides
- Motohiro Nonaka,
- Hideaki Mabashi-Asazuma,
- Donald L. Jarvis,
- Kazuhiko Yamasaki,
- Tomoya O. Akama,
- Masato Nagaoka,
- Toshio Sasai,
- Itsuko Kimura-Takagi,
- Yoichi Suwa,
- Takashi Yaegashi
- Published: January 6, 2021
- https://doi.org/10.1371/journal.pone.0241157