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Open Access
Peer-reviewed
Research Article
Preclinical evaluation of EPHX2 inhibition as a novel treatment for inflammatory bowel disease
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William C. Reisdorf ,
Contributed equally to this work with: William C. Reisdorf, Qing Xie
Roles Investigation, Visualization, Writing – original draft, Writing – review & editing
* E-mail: william.c.reisdorf@gsk.com
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Qing Xie ,
Contributed equally to this work with: William C. Reisdorf, Qing Xie
Roles Conceptualization, Formal analysis, Investigation, Resources, Visualization, Writing – original draft, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Xin Zeng,
Roles Formal analysis, Investigation, Writing – review & editing
Affiliation Target & Pathway Validation, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Wensheng Xie,
Roles Formal analysis, Investigation, Writing – review & editing
Affiliation Target & Pathway Validation, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Neetu Rajpal,
Roles Project administration, Resources, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Bao Hoang,
Roles Investigation, Resources, Writing – review & editing
Affiliation Exploratory Biomarkers, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Mark E. Burgert,
Roles Formal analysis, Writing – review & editing
Affiliation Research Statistics, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Vinod Kumar,
Roles Investigation, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Mark R. Hurle,
Roles Investigation, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Deepak K. Rajpal,
Roles Writing – original draft, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Sarah O’Donnell,
Roles Investigation, Writing – review & editing
Affiliation Centre for Digestive Diseases, Royal London Hospital, Barts Health NHS Trust, London, United Kingdom
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Thomas T. MacDonald,
Roles Conceptualization, Project administration, Supervision, Writing – review & editing
Affiliation Centre for Immunobiology, Blizard Institute, QMUL, London, United Kingdom
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Anna Vossenkämper,
Roles Investigation, Writing – review & editing
Affiliation Centre for Immunobiology, Blizard Institute, QMUL, London, United Kingdom
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Lin Wang,
Roles Investigation, Resources, Writing – review & editing
Affiliation Pattern Recognition Receptor DPU, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Mike Reilly,
Roles Conceptualization, Project administration, Supervision, Writing – review & editing
Affiliation Pattern Recognition Receptor DPU, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Bart J. Votta,
Roles Conceptualization, Project administration, Resources, Supervision, Writing – review & editing
Affiliation Pattern Recognition Receptor DPU, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Yolanda Sanchez,
Roles Conceptualization, Supervision, Writing – original draft, Writing – review & editing
Affiliation Stress and Repair DPU, Respiratory Therapy Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Pankaj Agarwal
Roles Conceptualization, Resources, Supervision, Writing – review & editing
Affiliation Computational Biology, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Preclinical evaluation of EPHX2 inhibition as a novel treatment for inflammatory bowel disease
- William C. Reisdorf,
- Qing Xie,
- Xin Zeng,
- Wensheng Xie,
- Neetu Rajpal,
- Bao Hoang,
- Mark E. Burgert,
- Vinod Kumar,
- Mark R. Hurle,
- Deepak K. Rajpal
- Published: April 19, 2019
- https://doi.org/10.1371/journal.pone.0215033