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Open Access
Peer-reviewed
Research Article
Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver
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Eric S. Muise ,
Contributed equally to this work with: Eric S. Muise, Hong-Ping Guan
Roles Conceptualization, Data curation, Formal analysis, Methodology, Visualization, Writing – original draft, Writing – review & editing
* E-mail: eric_muise@merck.com (ESM); iyassu@gmail.com (IKS)
Affiliation Genetics and Pharmacogenomics Department, MRL, Kenilworth, NJ, United States of America
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Hong-Ping Guan ,
Contributed equally to this work with: Eric S. Muise, Hong-Ping Guan
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Visualization, Writing – original draft, Writing – review & editing
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Jinqi Liu,
Roles Formal analysis, Investigation, Writing – original draft
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Andrea R. Nawrocki,
Roles Formal analysis, Methodology
Affiliation In Vivo Pharmacology Department, MRL, Kenilworth, NJ, United States of America
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Xiaodong Yang,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Chuanlin Wang,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Carlos G. Rodríguez,
Roles Investigation
Affiliation In Vivo Pharmacology Department, MRL, Kenilworth, NJ, United States of America
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Dan Zhou,
Roles Investigation
Affiliation In Vivo Pharmacology Department, MRL, Kenilworth, NJ, United States of America
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Judith N. Gorski,
Roles Investigation
Affiliation In Vivo Pharmacology Department, MRL, Kenilworth, NJ, United States of America
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Marc M. Kurtz,
Roles Investigation
Affiliation In Vitro PharmacologyDepartment, MRL, NJ, United States of America
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Danqing Feng,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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Kenneth J. Leavitt,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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Lan Wei,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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Robert R. Wilkening,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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James M. Apgar,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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Shiyao Xu,
Roles Investigation
Affiliation PPDM Preclinical ADME Department, MRL, Kenilworth, NJ, United States of America
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Ku Lu,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Wen Feng,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
⨯ -
Ying Li,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
⨯ -
Huaibing He,
Roles Investigation
Affiliation PPDM Preclinical ADME Department, MRL, Kenilworth, NJ, United States of America
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Stephen F. Previs,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
⨯ - Xiaolan Shen,
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Margaret van Heek,
Roles Supervision
Affiliation In Vivo Pharmacology Department, MRL, Kenilworth, NJ, United States of America
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Sandra C. Souza,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Mark J. Rosenbach,
Roles Investigation
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Tesfaye Biftu,
Roles Investigation
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
⨯ -
Mark D. Erion,
Roles Supervision
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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David E. Kelley,
Roles Conceptualization, Writing – original draft, Writing – review & editing
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Daniel M. Kemp,
Roles Conceptualization
Affiliation Biology-Discovery Department, MRL, Kenilworth, NJ, United States of America
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Robert W. Myers,
Roles Conceptualization, Formal analysis, Investigation, Methodology, Writing – original draft
Affiliation In Vitro PharmacologyDepartment, MRL, NJ, United States of America
⨯ - [ ... ],
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Iyassu K. Sebhat
Roles Conceptualization, Investigation, Writing – original draft, Writing – review & editing
* E-mail: eric_muise@merck.com (ESM); iyassu@gmail.com (IKS)
Affiliation Medicinal ChemistryDepartment, MRL, Kenilworth, NJ, United States of America
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Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver
- Eric S. Muise,
- Hong-Ping Guan,
- Jinqi Liu,
- Andrea R. Nawrocki,
- Xiaodong Yang,
- Chuanlin Wang,
- Carlos G. Rodríguez,
- Dan Zhou,
- Judith N. Gorski,
- Marc M. Kurtz
- Published: February 27, 2019
- https://doi.org/10.1371/journal.pone.0211568