Crystallographic and thermodynamic characterization of phenylaminopyridine bisphosphonates binding to human farnesyl pyrophosphate synthase

• Jaeok Park,

  Roles Conceptualization, Formal analysis, Investigation, Project administration, Resources, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing

  Affiliation Department of Biochemistry, McGill University, Montreal, Quebec, Canada

  http://orcid.org/0000-0002-8180-3950

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• Dmitry Rodionov,

  Roles Investigation

  Current address: Formulatrix, Bedford, Massachusetts, United States of America

  Affiliation Department of Biochemistry, McGill University, Montreal, Quebec, Canada

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• Joris W. De Schutter,

  Roles Resources

  Current address: Putnam Associates, Boston, Massachusetts, United States of America

  Affiliation Department of Chemistry, McGill University, Montreal, Quebec, Canada

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• Yih-Shyan Lin,

  Roles Resources

  Current address: APRINOIR Therapeutics, Taipei City, Taiwan

  Affiliation Department of Chemistry, McGill University, Montreal, Quebec, Canada

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• Youla S. Tsantrizos,

  Roles Conceptualization, Funding acquisition, Project administration, Supervision, Writing – review & editing

  Affiliations Department of Biochemistry, McGill University, Montreal, Quebec, Canada, Department of Chemistry, McGill University, Montreal, Quebec, Canada

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• Albert M. Berghuis

  Roles Conceptualization, Funding acquisition, Project administration, Supervision, Writing – review & editing

  * E-mail: albert.berghuis@mcgill.ca

  Affiliation Department of Biochemistry, McGill University, Montreal, Quebec, Canada

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