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Open Access
Peer-reviewed
Research Article
GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent
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Michele J. Pachanski,
Roles Data curation, Formal analysis, Methodology, Project administration, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Melissa E. Kirkland,
Roles Data curation, Formal analysis, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Daniel T. Kosinski,
Roles Data curation, Formal analysis, Investigation, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Joel Mane,
Roles Data curation, Investigation, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Boonlert Cheewatrakoolpong,
Roles Data curation, Formal analysis, Investigation, Methodology, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Jiyan Xue,
Roles Data curation, Formal analysis, Investigation, Methodology, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Daphne Szeto,
Roles Data curation, Formal analysis, Investigation, Methodology, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Gail Forrest,
Roles Data curation, Formal analysis, Methodology, Resources, Supervision, Validation
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Corin Miller,
Roles Investigation, Methodology, Supervision, Validation, Writing – original draft
Affiliation Translational Imaging Biomarkers, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Michelle Bunzel,
Roles Investigation, Methodology, Validation
Affiliation Translational Imaging Biomarkers, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Christopher W. Plummer,
Roles Resources
Affiliation Department of Medicinal Chemistry, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Harry R. Chobanian,
Roles Conceptualization, Resources, Writing – review & editing
Affiliation Department of Medicinal Chemistry, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Michael W. Miller,
Roles Project administration, Resources
Affiliation Department of Medicinal Chemistry, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Sarah Souza,
Roles Data curation, Investigation, Methodology, Validation
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Brande S. Thomas-Fowlkes,
Roles Data curation, Investigation, Methodology, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Aimie M. Ogawa,
Roles Data curation, Investigation, Methodology, Validation, Visualization
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Adam B. Weinglass,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Jerry Di Salvo,
Roles Conceptualization, Formal analysis, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Xiaoyan Li,
Roles Conceptualization, Methodology, Resources, Supervision, Visualization, Writing – review & editing
Affiliation Department of Cardio Metabolic Diseases, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Yue Feng,
Roles Investigation, Methodology, Resources, Validation, Visualization
Affiliation Department of Cardio Metabolic Diseases, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Daniel A. Tatosian,
Roles Conceptualization, Formal analysis, Methodology, Visualization, Writing – original draft, Writing – review & editing
Affiliation Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Andrew D. Howard,
Roles Project administration, Resources, Supervision
Affiliation Department of Cardio Metabolic Diseases, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Steven L. Colletti,
Roles Project administration, Resources, Supervision, Writing – review & editing
Affiliation Department of Medicinal Chemistry, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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Maria E. Trujillo
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
* E-mail: maria_trujillo@merck.com
Affiliation In Vivo Pharmacology, Merck & Co., Inc., Kenilworth, New Jersey, United States of America
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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent
- Michele J. Pachanski,
- Melissa E. Kirkland,
- Daniel T. Kosinski,
- Joel Mane,
- Boonlert Cheewatrakoolpong,
- Jiyan Xue,
- Daphne Szeto,
- Gail Forrest,
- Corin Miller,
- Michelle Bunzel
- Published: October 20, 2017
- https://doi.org/10.1371/journal.pone.0186033