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Open Access
Peer-reviewed
Research Article
Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-care
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Kathleen M. Gillooly,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Visualization, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Claudine Pulicicchio,
Roles Data curation, Investigation, Methodology, Visualization, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Mark A. Pattoli,
Roles Data curation, Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Lihong Cheng,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Stacey Skala,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Elizabeth M. Heimrich,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Kim W. McIntyre,
Roles Conceptualization, Data curation, Formal analysis, Methodology, Project administration, Supervision, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Tracy L. Taylor,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Daniel W. Kukral,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Exploratory Clinical and Translational Research, Imaging, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Shailesh Dudhgaonkar,
Roles Formal analysis, Resources, Supervision, Writing – review & editing
Affiliation Disease Sciences and Technology, Biocon Bristol-Myers Squibb Research Center, Syngene International Limited, Bangalore, India
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Jignesh Nagar,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Disease Sciences and Technology, Biocon Bristol-Myers Squibb Research Center, Syngene International Limited, Bangalore, India
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Dana Banas,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Discovery Translational Sciences, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Scott H. Watterson,
Roles Investigation, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Chemistry, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Joseph A. Tino,
Roles Conceptualization, Methodology, Writing – review & editing
Affiliation Immunosciences Discovery Chemistry, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Aberra Fura,
Roles Conceptualization, Project administration, Writing – review & editing
Affiliation Department of Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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James R. Burke
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing
* E-mail: james.burke@bms.com
Affiliation Immunosciences Discovery Biology, Bristol-Myers Squibb Research & Development, Princeton, New Jersey, United States of America
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Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-care
- Kathleen M. Gillooly,
- Claudine Pulicicchio,
- Mark A. Pattoli,
- Lihong Cheng,
- Stacey Skala,
- Elizabeth M. Heimrich,
- Kim W. McIntyre,
- Tracy L. Taylor,
- Daniel W. Kukral,
- Shailesh Dudhgaonkar
- Published: July 24, 2017
- https://doi.org/10.1371/journal.pone.0181782