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Open Access
Peer-reviewed
Research Article
Discovery and Molecular Basis of a Diverse Set of Polycomb Repressive Complex 2 Inhibitors Recognition by EED
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Ling Li ,
Contributed equally to this work with: Ling Li, Hailong Zhang
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Hailong Zhang ,
Contributed equally to this work with: Ling Li, Hailong Zhang
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Man Zhang,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Mengxi Zhao,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Lijian Feng,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Xiao Luo,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Zhenting Gao,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Ying Huang,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Ophelia Ardayfio,
Affiliation Novartis Institutes for BioMedical Research, Cambridge, Massachusetts, United States of America
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Ji-Hu Zhang,
Affiliation Novartis Institutes for BioMedical Research, Cambridge, Massachusetts, United States of America
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Ying Lin,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Hong Fan,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Yuan Mi,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Guobin Li,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Lei Liu,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Leying Feng,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Fangjun Luo,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Lin Teng,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Wei Qi,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Johannes Ottl,
Affiliation Novartis Institutes for BioMedical Research, Basel, Switzerland
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Andreas Lingel,
Affiliation Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Dirksen E. Bussiere,
Affiliation Novartis Institutes for BioMedical Research, Emeryville, California, United States of America
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Zhengtian Yu,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Peter Atadja,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Chris Lu,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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En Li,
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Justin Gu ,
* E-mail: Kehao.zhao@novartis.com (KZ); Justin.gu@novartis.com (JG)
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
⨯ - [ ... ],
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Kehao Zhao
* E-mail: Kehao.zhao@novartis.com (KZ); Justin.gu@novartis.com (JG)
Affiliation China Novartis Institutes for BioMedical Research, Shanghai, China
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Discovery and Molecular Basis of a Diverse Set of Polycomb Repressive Complex 2 Inhibitors Recognition by EED
- Ling Li,
- Hailong Zhang,
- Man Zhang,
- Mengxi Zhao,
- Lijian Feng,
- Xiao Luo,
- Zhenting Gao,
- Ying Huang,
- Ophelia Ardayfio,
- Ji-Hu Zhang
- Published: January 10, 2017
- https://doi.org/10.1371/journal.pone.0169855