Effect of BET Missense Mutations on Bromodomain Function, Inhibitor Binding and Stability

• Laura Lori,

  Affiliation Department of Biochemical Sciences “A. Rossi Fanelli”, Sapienza University of Rome, Rome, Italy

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• Alessandra Pasquo,

  Affiliation SSPT-BIOAG-BIOTEC ENEA Casaccia ENEA, Rome, Italy

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• Clorinda Lori,

  Affiliation Department of Biochemical Sciences “A. Rossi Fanelli”, Sapienza University of Rome, Rome, Italy

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• Maria Petrosino,

  Affiliation Department of Biochemical Sciences “A. Rossi Fanelli”, Sapienza University of Rome, Rome, Italy

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• Roberta Chiaraluce ,

  * E-mail: roberta.chiaraluce@uniroma1.it

  Affiliation Department of Biochemical Sciences “A. Rossi Fanelli”, Sapienza University of Rome, Rome, Italy

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• Cynthia Tallant,

  Current address: Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences (BMLS), Johann Wolfgang Goethe-University, Frankfurt am Main, Germany

  Affiliation Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute, University of Oxford, Oxford, United Kingdom

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• Stefan Knapp,

  Current address: Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences (BMLS), Johann Wolfgang Goethe-University, Frankfurt am Main, Germany

  Affiliation Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute, University of Oxford, Oxford, United Kingdom

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• Valerio Consalvi

  Affiliation Department of Biochemical Sciences “A. Rossi Fanelli”, Sapienza University of Rome, Rome, Italy

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