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Open Access
Peer-reviewed
Research Article
A Novel Triazolopyridine-Based Spleen Tyrosine Kinase Inhibitor That Arrests Joint Inflammation
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Gregory D. Ferguson ,
* E-mail: gferguson66@yahoo.com
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Mercedes Delgado,
Affiliation Department of Chemistry, Celgene Corporation, San Diego, California, United States of America
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Veronique Plantevin-Krenitsky,
Affiliation Department of Chemistry, Celgene Corporation, San Diego, California, United States of America
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Kristen Jensen-Pergakes,
Affiliation Department of Tumor Cell Biology, Pfizer Corporation, San Diego, California, United States of America
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R. J. Bates,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Sanaa Torres,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Maria Celeridad,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Heather Brown,
Affiliation Department of Pharmacology, Celgene Corporation, San Diego, California, United States of America
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Kelven Burnett,
Affiliation Department of Pharmacology, Celgene Corporation, San Diego, California, United States of America
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Lisa Nadolny,
Affiliation Department of Chemistry, Celgene Corporation, San Diego, California, United States of America
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Lida Tehrani,
Affiliation Department of Chemistry, Celgene Corporation, San Diego, California, United States of America
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Garrick Packard,
Affiliation Department of Chemistry, Celgene Corporation, San Diego, California, United States of America
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Barbra Pagarigan,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Jason Haelewyn,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Trish Nguyen,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Li Xu,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Yang Tang,
Affiliation Department of Pharmacology, Celgene Corporation, San Diego, California, United States of America
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Matthew Hickman,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Frans Baculi,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Steven Pierce,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Keiji Miyazawa,
Affiliation Department of Corporate Planning and Strategy, Kissei Pharmaceutical Company, Matsumoto City, Nagano, Japan
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Pilgrim Jackson,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Philip Chamberlain,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Laurie LeBrun,
Affiliation Department of Biochemistry, Celgene Corporation, San Diego, California, United States of America
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Weilin Xie,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Brydon Bennett,
Affiliation Department of Inflammation Research, Celgene Corporation, San Diego, California, United States of America
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Kate Blease
Affiliation Department of Pharmacology, Celgene Corporation, San Diego, California, United States of America
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A Novel Triazolopyridine-Based Spleen Tyrosine Kinase Inhibitor That Arrests Joint Inflammation
- Gregory D. Ferguson,
- Mercedes Delgado,
- Veronique Plantevin-Krenitsky,
- Kristen Jensen-Pergakes,
- R. J. Bates,
- Sanaa Torres,
- Maria Celeridad,
- Heather Brown,
- Kelven Burnett,
- Lisa Nadolny
- Published: January 12, 2016
- https://doi.org/10.1371/journal.pone.0145705