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Open Access
Peer-reviewed
Research Article
Identification of Novel Small Molecule Inhibitors of Oncogenic RET Kinase
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Marialuisa Moccia,
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Qingsong Liu,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Teresa Guida,
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Giorgia Federico,
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Annalisa Brescia,
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Zheng Zhao,
Affiliation High Magnetic Field Laboratory, Chinese Academy of Sciences, Hefei, Anhui, P.R. China
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Hwan Geun Choi,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Xianming Deng,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Li Tan,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Jinhua Wang,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Marc Billaud,
Affiliation Institut Albert Bonniot, CRI INSERM/UJF U823, La Tronche Cedex, France
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Nathanael S. Gray,
Affiliations Department of Cancer Biology, Dana Farber Cancer Institute, Boston, Massachusetts United States of America, Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America
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Francesca Carlomagno ,
Contributed equally to this work with: Francesca Carlomagno, Massimo Santoro
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Massimo Santoro
Contributed equally to this work with: Francesca Carlomagno, Massimo Santoro
* E-mail: masantor@unina.it
Affiliations Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Università di Napoli “Federico II”, Naples, Italy, Istituto di Endocrinologia ed Oncologia Sperimentale del CNR, Naples, Italy
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Identification of Novel Small Molecule Inhibitors of Oncogenic RET Kinase
- Marialuisa Moccia,
- Qingsong Liu,
- Teresa Guida,
- Giorgia Federico,
- Annalisa Brescia,
- Zheng Zhao,
- Hwan Geun Choi,
- Xianming Deng,
- Li Tan,
- Jinhua Wang
- Published: June 5, 2015
- https://doi.org/10.1371/journal.pone.0128364