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Open Access
Peer-reviewed
Research Article
MCL1 and BCL-xL Levels in Solid Tumors Are Predictive of Dinaciclib-Induced Apoptosis
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Robert N. Booher,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Harold Hatch,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Brian M. Dolinski,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Thi Nguyen,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Lauren Harmonay,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Ali-Samer Al-Assaad,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Mark Ayers,
Affiliation BioInformatics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Michael Nebozhyn,
Affiliation BioInformatics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Andrey Loboda,
Affiliation BioInformatics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Heather A. Hirsch,
Affiliation BioInformatics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Theresa Zhang,
Affiliation BioInformatics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Bin Shi,
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Carrie E. Merkel,
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Minilik H. Angagaw,
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Yaolin Wang,
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Brian J. Long,
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Xianlu Q. Lennon,
Affiliation Biomarkers, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Nathan Miselis,
Affiliation Biomarkers, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Vincenzo Pucci,
Affiliation Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck Research Laboratories, Boston, Massachusetts, United States of America
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James W. Monahan,
Affiliation Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Junghoon Lee,
Affiliation Quantitative Pharmacology and Pharmacometrics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Anna Georgieva Kondic,
Affiliation Quantitative Pharmacology and Pharmacometrics, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Eun Kyung Im,
Affiliation Clinical Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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David Mauro,
Affiliation Clinical Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Rebecca Blanchard,
Affiliation Clinical Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Gary Gilliland,
Affiliation Clinical Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Stephen E. Fawell,
Current address: AstraZeneca, Waltham, Massachusetts, United States of America
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Leigh Zawel,
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Alwin G. Schuller,
Current address: AstraZeneca, Waltham, Massachusetts, United States of America
Affiliation In vivo Pharmacology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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Peter Strack
* E-mail: cpstrack@verizon.net
Affiliation Discovery Oncology, Merck Research Laboratories, Boston, Massachusetts, United States of America
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MCL1 and BCL-xL Levels in Solid Tumors Are Predictive of Dinaciclib-Induced Apoptosis
- Robert N. Booher,
- Harold Hatch,
- Brian M. Dolinski,
- Thi Nguyen,
- Lauren Harmonay,
- Ali-Samer Al-Assaad,
- Mark Ayers,
- Michael Nebozhyn,
- Andrey Loboda,
- Heather A. Hirsch
- Published: October 7, 2014
- https://doi.org/10.1371/journal.pone.0108371