De Novo Peptide Design and Experimental Validation of Histone Methyltransferase Inhibitors

• James Smadbeck,

  Affiliation Department of Chemical and Biological Engineering, Princeton University, Princeton, New Jersey, United States of America

  ⨯
• Meghan B. Peterson,

  Affiliation Department of Chemical and Biological Engineering, Princeton University, Princeton, New Jersey, United States of America

  ⨯
• Barry M. Zee,

  Affiliation Department of Molecular Biology, Princeton University, Princeton, New Jersey, United States of America

  ⨯
• Shivani Garapaty,

  Affiliation Constellation Pharmaceuticals, Cambridge, Massachusetts, United States of America

  ⨯
• Aashna Mago,

  Affiliation Department of Molecular Biology, Princeton University, Princeton, New Jersey, United States of America

  ⨯
• Christina Lee,

  Affiliation Constellation Pharmaceuticals, Cambridge, Massachusetts, United States of America

  ⨯
• Athanassios Giannis,

  Affiliation University of Leipzig, Institute of Organic Chemistry, Leipzig, Germany

  ⨯
• Patrick Trojer,

  Affiliation Constellation Pharmaceuticals, Cambridge, Massachusetts, United States of America

  ⨯
• Benjamin A. Garcia,

  Affiliations Department of Molecular Biology, Princeton University, Princeton, New Jersey, United States of America, Department of Chemistry, Princeton University, Princeton, New Jersey, United States of America, Epigenetics Program, Department of Biochemistry and Biophysics, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America

  ⨯
• Christodoulos A. Floudas

  * E-mail: floudas@titan.princeton.edu

  Affiliation Department of Chemical and Biological Engineering, Princeton University, Princeton, New Jersey, United States of America

  ⨯