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Open Access
Peer-reviewed
Research Article
Identification of Benzimidazole Diamides as Selective Inhibitors of the Nucleotide-Binding Oligomerization Domain 2 (NOD2) Signaling Pathway
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David J. Rickard ,
* E-mail: David.J.Rickard@gsk.com
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Clark A. Sehon,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Viera Kasparcova,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Lorena A. Kallal,
Affiliation Biological Reagents and Assay Development, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Xin Zeng,
Affiliation Screening and Compound Profiling, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Monica N. Montoute,
Affiliation Screening and Compound Profiling, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Tushar Chordia,
Affiliation Biological Reagents and Assay Development, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Derek D. Poore,
Affiliation Biological Reagents and Assay Development, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Hu Li,
Affiliation Biological Reagents and Assay Development, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Zining Wu,
Affiliation Screening and Compound Profiling, Platform Technology Sciences, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Patrick M. Eidam,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Pamela A. Haile,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Jong Yu,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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John G. Emery,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Robert W. Marquis,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Peter J. Gough,
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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John Bertin
Affiliation Pattern Recognition Receptor Discovery Performance Unit, Immuno-Inflammation Therapeutic Area, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America
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Identification of Benzimidazole Diamides as Selective Inhibitors of the Nucleotide-Binding Oligomerization Domain 2 (NOD2) Signaling Pathway
- David J. Rickard,
- Clark A. Sehon,
- Viera Kasparcova,
- Lorena A. Kallal,
- Xin Zeng,
- Monica N. Montoute,
- Tushar Chordia,
- Derek D. Poore,
- Hu Li,
- Zining Wu
- Published: August 1, 2013
- https://doi.org/10.1371/journal.pone.0069619