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Open Access
Peer-reviewed
Research Article
Application of Multiplexed Kinase Inhibitor Beads to Study Kinome Adaptations in Drug-Resistant Leukemia
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Matthew J. Cooper,
Affiliations Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America, Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America, Curriculum in Genetics & Molecular Biology, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Nathan J. Cox,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Eric I. Zimmerman,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Brian J. Dewar,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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James S. Duncan,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Martin C. Whittle,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Thien A. Nguyen,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Lauren S. Jones,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Sreerupa Ghose Roy,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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David M. Smalley,
Affiliation Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Pei Fen Kuan,
Affiliations Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America, Department of Biostatistics, Gillings School of Global Public Health, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Kristy L. Richards,
Affiliations Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America, Division of Hematology & Oncology, Department of Medicine, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Richard I. Christopherson,
Affiliation School of Molecular Bioscience, University of Sydney, Sydney, New South Wales, Australia
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Jian Jin,
Affiliation Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Stephen V. Frye,
Affiliation Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Gary L. Johnson,
Affiliations Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America, Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Albert S. Baldwin,
Affiliations Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America, Curriculum in Genetics & Molecular Biology, University of North Carolina, Chapel Hill, North Carolina, United States of America, Department of Biology, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Lee M. Graves
* E-mail: lmg@med.unc.edu
Affiliations Department of Pharmacology, School of Medicine, University of North Carolina, Chapel Hill, North Carolina, United States of America, Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, North Carolina, United States of America
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Application of Multiplexed Kinase Inhibitor Beads to Study Kinome Adaptations in Drug-Resistant Leukemia
- Matthew J. Cooper,
- Nathan J. Cox,
- Eric I. Zimmerman,
- Brian J. Dewar,
- James S. Duncan,
- Martin C. Whittle,
- Thien A. Nguyen,
- Lauren S. Jones,
- Sreerupa Ghose Roy,
- David M. Smalley
- Published: June 24, 2013
- https://doi.org/10.1371/journal.pone.0066755