A Targeted Library Screen Reveals a New Inhibitor Scaffold for Protein Kinase D

Open Access

Peer-reviewed

Research Article

Manuj Tandon ,

Contributed equally to this work with: Manuj Tandon, Lirong Wang

Affiliation Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America
⨯
Lirong Wang ,

Contributed equally to this work with: Manuj Tandon, Lirong Wang

Affiliation Department of Pharmaceutical Sciences, University of Pittsburgh, Pittsburgh, Pennsylavania, United States of America
⨯
Qi Xu,

Affiliation Department of Pharmaceutical Sciences, University of Pittsburgh, Pittsburgh, Pennsylavania, United States of America
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Xiangqun Xie,

Affiliation Department of Pharmaceutical Sciences, University of Pittsburgh, Pittsburgh, Pennsylavania, United States of America
⨯
Peter Wipf ,

* E-mail: pwipf@pitt.edu (PW); qjw1@pitt.edu (QJW)

Affiliations Department of Chemistry and Center for Chemical Methodologies and Library Development, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmaceutical Sciences, University of Pittsburgh, Pittsburgh, Pennsylavania, United States of America
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Qiming Jane Wang

* E-mail: pwipf@pitt.edu (PW); qjw1@pitt.edu (QJW)

Affiliation Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America
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In vitro kinase assay
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Protein kinases
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Small molecules
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