About the Authors

James F. Sampson

Roles Conceptualization, Data curation, Formal analysis, Investigation, Project administration, Writing – original draft

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Hong Zhang

Roles Conceptualization, Data curation, Investigation, Methodology, Validation, Writing – review & editing

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Dongmei Zhang

Roles Data curation, Investigation, Validation, Writing – review & editing

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Mingying Bi

Roles Investigation

Affiliation Discovery R and D, Teva Pharmaceutical Industries, Ltd., Redwood City, United States of America

Adam Hinthorne

Roles Data curation, Investigation, Methodology, Project administration, Resources

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Sakeena Syed

Roles Data curation, Investigation, Methodology, Project administration, Resources

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Yuhong Zhang

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – review & editing

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Nibedita Chattopadhyay

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Sabrina Collins

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Sarah Pogue

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing

Affiliation Discovery R and D, Teva Pharmaceutical Industries, Ltd., Redwood City, United States of America

Pia Björck

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Writing – original draft, Writing – review & editing

Affiliation Discovery R and D, Teva Pharmaceutical Industries, Ltd., Redwood City, United States of America

Michael Curley

Roles Conceptualization, Investigation, Methodology, Project administration, Supervision, Writing – original draft, Writing – review & editing

michael.curley@takeda.com

Affiliation Oncology Drug Discovery Unit, Takeda Development Center Americas, Inc. (TDCA), Lexington, Massachusetts, United States of America

Competing Interests

J.F.S. reports employment with Takeda. H.Z. reports employment with Takeda at the time of the study. D.Z. reports employment with Takeda. M.B. reports employment with Teva. A.H. reports employment with Takeda. S.S. reports employment with Takeda at the time of the study. Y.Z. reports employment with and ownership of stock/shares in Takeda. N.C. reports employment with Takeda at the time of the study. S.C. reports employment with and ownership of stock/shares in Takeda. S.P. and P.B. report employment with and ownership of stock/shares in Teva. M.C. reports employment with and ownership of stock/shares in Takeda, and ownership of stock/shares in Merrimack Pharmaceuticals.