About the Authors

Archana Bommi-Reddy

Contributed equally to this work with: Archana Bommi-Reddy, Sungmi Park-Chouinard, David N. Mayhew

Roles Conceptualization, Formal analysis, Investigation, Project administration, Writing – original draft

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Sungmi Park-Chouinard

Contributed equally to this work with: Archana Bommi-Reddy, Sungmi Park-Chouinard, David N. Mayhew

Roles Conceptualization, Formal analysis, Investigation, Visualization, Writing – original draft

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

David N. Mayhew

Contributed equally to this work with: Archana Bommi-Reddy, Sungmi Park-Chouinard, David N. Mayhew

Roles Data curation, Formal analysis, Software, Visualization, Writing – original draft

Current address: Foghorn Therapeutics, Cambridge, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Esteban Terzo

Roles Investigation

Current address: Eloxx Pharmaceuticals, Watertown, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Aparna Hingway

Roles Investigation

Current address: Novartis Institutes for Biomedical Research, Cambridge, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Michael J. Steinbaugh

Roles Formal analysis, Software

Current address: 28–7 Therapeutics, Cambridge, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Jonathan E. Wilson

Roles Conceptualization, Project administration

Current address: Flare Therapeutics, Cambridge, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Robert J. Sims III

Roles Conceptualization, Project administration

Current address: Flare Therapeutics, Cambridge, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Andrew R. Conery

Roles Conceptualization, Formal analysis, Visualization, Writing – original draft

arconery@gmail.com

Current address: Triana Biomedicines, Waltham, Massachusetts, United States of America

Affiliation Constellation Pharmaceuticals, a Morphosys Company, Cambridge, Massachusetts, United States of America

Competing Interests

Authors are current or former employees and stockholders of Constellation Pharmaceuticals, a Morphosys company, which provided funding for this research. Patents have been filed around the chemical series that includes CPI-1612. This work does not relate to any marketed products or products in development. These disclosures do not alter our adherence to PLOS ONE policies on sharing data and materials.