About the Authors

Michael R. Weed

Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing

mweed@rx-gen.com

Current address: CNS Disease and Physiology, RxGen, Inc., New Haven, CT, United States of America

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Joseph Polino

Roles Data curation, Investigation, Methodology, Project administration, Supervision, Validation, Writing – original draft, Writing – review & editing

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Laura Signor

Roles Data curation, Investigation, Methodology

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Mark Bookbinder

Roles Data curation, Investigation

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Deborah Keavy

Roles Investigation

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Yulia Benitex

Roles Data curation, Investigation

Affiliation Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Daniel G. Morgan

Roles Data curation, Investigation, Resources, Supervision

Affiliation Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Dalton King

Roles Investigation, Resources, Writing – review & editing

Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

John E. Macor

Roles Conceptualization, Resources, Supervision

Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Robert Zaczek

Roles Conceptualization, Resources, Supervision

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Richard Olson

Roles Conceptualization, Resources, Supervision

Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Linda J. Bristow

Roles Conceptualization, Resources, Supervision, Writing – review & editing

Affiliation Genetically Defined Diseases and Genomics, Bristol-Myers Squibb Company, Wallingford, CT, United States of America

Competing Interests

All authors were employees of Bristol-Myers Squibb during these studies, and some authors own stock in BMS. The authors have declared that no competing interests exist. This does not alter the authors' adherence to PLOS ONE policies on sharing data and materials.