About the Authors
- Linda J. Bristow
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* E-mail: Linda.bristow@bms.com
Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Amy E. Easton
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Yu-Wen Li
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Digavalli V. Sivarao
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Regina Lidge
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Kelli M. Jones
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Debra Post-Munson
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Christopher Daly
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Nicholas J. Lodge
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Lizbeth Gallagher
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Affiliation Lead Discovery and Optimization, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Thaddeus Molski
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Richard Pieschl
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Ping Chen
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Adam Hendricson
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Affiliation Lead Discovery and Optimization, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Ryan Westphal
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- James Cook
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Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Christiana Iwuagwu
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Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Daniel Morgan
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Affiliation Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Yulia Benitex
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Affiliation Pharmaceutical Candidate Optimization, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Dalton King
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Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- John E. Macor
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Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Robert Zaczek
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Affiliation Discovery Biology, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
- Richard Olson
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Affiliation Discovery Chemistry, Bristol-Myers Squibb Company, Wallingford, Connecticut, United States of America
Competing Interests
All authors were paid employees of Bristol-Myers Squibb Company at the time this research was conducted. In addition many authors own Bristol-Myers Squibb Company stock and some are inventors on patents relating to BMS-933043, the agent described in this manuscript. This does not alter the authors' adherence to PLOS ONE policies on sharing data and materials.
Author Contributions
Conceived and designed the experiments: LJB AEE Y-WL DVS NJL RW DM DK JEM RZ RO. Performed the experiments: RL KMJ DP-M CD LG TM RP PC AH JC CI YB. Analyzed the data: AAEE Y-WL DVS RL KMJ DP-M CD NJL LG TM RP PC AH RW DM YB. Contributed reagents/materials/analysis tools: JC CI DK. Wrote the paper: LJB.