About the Authors
- Yonchu Jenkins
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Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Tian-Qiang Sun
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Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Vadim Markovtsov
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Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Marc Foretz
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Affiliations Inserm, U1016, Institut Cochin, Paris, France, CNRS, UMR8104, Paris, France, Université Paris Descartes, Sorbonne Paris cité, Paris, France
- Wei Li
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Henry Nguyen
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Yingwu Li
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Alison Pan
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Gerald Uy
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Lisa Gross
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Kristen Baltgalvis
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Stephanie L. Yung
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Tarikere Gururaja
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Taisei Kinoshita
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Alexander Owyang
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Ira J. Smith
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Kelly McCaughey
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Kathy White
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Guillermo Godinez
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Raniel Alcantara
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Carmen Choy
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Hong Ren
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Rachel Basile
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- David J. Sweeny
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Xiang Xu
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Sarkiz D. Issakani
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- David C. Carroll
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Dane A. Goff
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Simon J. Shaw
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Rajinder Singh
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Laszlo G. Boros
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Affiliations SiDMAP, LLC, Los Angeles, California, United States of America, Department of Pediatrics, Los Angeles Biomedical Research Institute (LABIOMED) at the Harbor-UCLA Medical Center, Torrance, California, United States of America
- Marc-André Laplante
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Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
- Bruno Marcotte
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Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
- Rita Kohen
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Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
- Benoit Viollet
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Affiliations Inserm, U1016, Institut Cochin, Paris, France, CNRS, UMR8104, Paris, France, Université Paris Descartes, Sorbonne Paris cité, Paris, France
- André Marette
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Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
- Donald G. Payan
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Todd M. Kinsella
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Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
- Yasumichi Hitoshi
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* E-mail: yhitoshi@rigel.com
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
Competing Interests
YJ, TQS, VM, WL, HN, YL, AP, GU, LG, KB, SLY, TG, TK, AO, IJS, KM, KW, GG, RA, CC, HR, RB, DJS, XX, SDI, DCC, DAG, SJS, RS, DGP, TMK and YH are or have been employees of Rigel Pharmaceuticals, Inc. LGB is an employee of SiDMAP, LLC. The remaining authors declare no competing financial interests. This does not alter the authors' adherence to all the PLOS ONE policies on sharing data and materials.
Author Contributions
Conceived and designed the experiments: YJ VM TQS TMK DPG YH. Performed the experiments: YJ VM TQS TMK YH WQL MF BV HN YL AP GU LG KB SLY TG TK AO IJS KM KW GG RA CC HR RB DJS XX SDI DCC DAG SJS RS LGB MAL BM RK AM. Analyzed the data: YJ VM TQS TMK YH WQL MF BV HN YL AP GU LG KB SLY TG TK AO IJS KM KW GG RA CC HR RB DJS XX SDI DCC DAG SJS RS LGB MAL BM RK AM. Contributed reagents/materials/analysis tools: DCC DAG SJS RS. Wrote the manuscript: YJ VM TQS TMK WQL DGP AM YH.