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Open Access
Peer-reviewed
Research Article
Progress towards a public chemogenomic set for protein kinases and a call for contributions
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David H. Drewry ,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: David.Drewry@unc.edu
Affiliation Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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Carrow I. Wells,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Visualization, Writing – original draft, Writing – review & editing
Affiliation Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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David M. Andrews,
Roles Conceptualization
Affiliation AstraZeneca, Darwin Building, Cambridge Science Park, Cambridge, United Kingdom
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Richard Angell,
Roles Conceptualization, Writing – review & editing
Affiliation Drug Discovery Group, Translational Research Office, University College London School of Pharmacy, 29–39 Brunswick Square, London, United Kingdom
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Hassan Al-Ali,
Roles Conceptualization, Formal analysis, Methodology, Writing – review & editing
Affiliations Miami Project to Cure Paralysis, University of Miami Miller School of Medicine, Miami, Florida, United States of America, Peggy and Harold Katz Family Drug Discovery Center, University of Miami Miller School of Medicine, Miami, Florida, United States of America
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Alison D. Axtman,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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Stephen J. Capuzzi,
Roles Formal analysis, Writing – original draft
Affiliation Laboratory for Molecular Modeling, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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Jonathan M. Elkins,
Roles Conceptualization, Writing – review & editing
Affiliation Structural Genomics Consortium, Universidade Estadual de Campinas—UNICAMP, Campinas, Sao Paulo, Brazil
⨯ - Peter Ettmayer,
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Mathias Frederiksen,
Roles Conceptualization
Affiliation Novartis Institutes for BioMedical Research, Novartis Campus, Basel, Switzerland
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Opher Gileadi,
Roles Conceptualization, Writing – review & editing
Affiliation Structural Genomics Consortium and Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford, United Kingdom
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Nathanael Gray,
Roles Conceptualization
Affiliations Harvard Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, United States of America, Department of Cancer Biology, Dana−Farber Cancer Institute, Boston, Massachusetts, United States of America
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Alice Hooper,
Roles Conceptualization, Data curation, Formal analysis
Affiliation Drug Discovery Group, Translational Research Office, University College London School of Pharmacy, 29–39 Brunswick Square, London, United Kingdom
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Stefan Knapp,
Roles Conceptualization, Writing – review & editing
Affiliation Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, and Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, Max-von-Laue-Straße 15, Frankfurt am Main, Germany
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Stefan Laufer,
Roles Conceptualization
Affiliation Department of Pharmaceutical Chemistry, Institute of Pharmaceutical Sciences, Eberhard Karls Universität Tübingen, Auf der Morgenstelle 8, Tübingen, Germany
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Ulrich Luecking,
Roles Conceptualization
Affiliation Bayer Pharma AG, Drug Discovery, Müllerstrasse 178, Berlin, Germany
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Michael Michaelides,
Roles Conceptualization
Affiliation Oncology Chemistry, AbbVie, 1 North Waukegan Road, North Chicago, Illinois, United States of America
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Susanne Müller,
Roles Conceptualization, Writing – review & editing
Affiliation Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, and Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, Max-von-Laue-Straße 15, Frankfurt am Main, Germany
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Eugene Muratov,
Roles Formal analysis
Affiliation Laboratory for Molecular Modeling, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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R. Aldrin Denny,
Roles Conceptualization
Affiliation Worldwide Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts, United States of America
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Kumar S. Saikatendu,
Roles Conceptualization
Affiliation Global Research Externalization, Takeda California, Inc., 10410 Science Center Drive, San Diego, California, United States of America
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Daniel K. Treiber,
Roles Formal analysis, Visualization, Writing – review & editing
Affiliation DiscoverX Corporation,Fremont, California, United States of America
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William J. Zuercher,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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Timothy M. Willson
Roles Conceptualization, Supervision, Writing – original draft, Writing – review & editing
Affiliation Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, United States of America
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Progress towards a public chemogenomic set for protein kinases and a call for contributions
- David H. Drewry,
- Carrow I. Wells,
- David M. Andrews,
- Richard Angell,
- Hassan Al-Ali,
- Alison D. Axtman,
- Stephen J. Capuzzi,
- Jonathan M. Elkins,
- Peter Ettmayer,
- Mathias Frederiksen
- Published: August 2, 2017
- https://doi.org/10.1371/journal.pone.0181585
- See the preprint