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Evaluation of robenidine analog NCL195 as a novel broad-spectrum antibacterial agent

  • Abiodun D. Ogunniyi ,

    Contributed equally to this work with: Abiodun D. Ogunniyi, Manouchehr Khazandi, Andrew J. Stevens

    Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Supervision, Validation, Writing – original draft, Writing – review & editing

    david.ogunniyi@adelaide.edu.au (ADO); darren.trott@adelaide.edu.au (DJT)

    Affiliation Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Manouchehr Khazandi ,

    Contributed equally to this work with: Abiodun D. Ogunniyi, Manouchehr Khazandi, Andrew J. Stevens

    Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Writing – original draft, Writing – review & editing

    Affiliation Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Andrew J. Stevens ,

    Contributed equally to this work with: Abiodun D. Ogunniyi, Manouchehr Khazandi, Andrew J. Stevens

    Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Writing – original draft, Writing – review & editing

    Affiliation Chemistry, School of Environmental & Life Sciences, The University of Newcastle, Callaghan, New South Wales, Australia

  • Sarah K. Sims,

    Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Validation, Writing – original draft, Writing – review & editing

    Affiliation School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Stephen W. Page,

    Roles Conceptualization, Formal analysis, Funding acquisition, Resources, Writing – review & editing

    Affiliation Neoculi Pty Ltd, Burwood, Victoria, Australia

  • Sanjay Garg,

    Roles Conceptualization, Formal analysis, Methodology, Resources, Supervision, Writing – review & editing

    Affiliation Centre for Pharmaceutical Innovation and Development, School of Pharmacy and Medical Sciences, Sansom Institute for Health Research, University of South Australia, Adelaide, South Australia, Australia

  • Henrietta Venter,

    Roles Conceptualization, Formal analysis, Funding acquisition, Investigation, Methodology, Resources, Writing – review & editing

    Affiliation School of Pharmacy and Medical Sciences, Sansom Institute for Health Research, University of South Australia, Adelaide, South Australia, Australia

  • Andrew Powell,

    Roles Data curation, Formal analysis, Investigation, Project administration, Writing – review & editing

    Affiliation Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia

  • Karen White,

    Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Supervision, Writing – review & editing

    Affiliation Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia

  • Kiro R. Petrovski,

    Roles Formal analysis, Funding acquisition, Writing – review & editing

    Affiliation Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Geraldine Laven-Law,

    Roles Conceptualization, Data curation, Investigation, Methodology, Writing – review & editing

    Affiliation School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Eliane G. Tótoli,

    Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Writing – review & editing

    Affiliation Department of Drugs and Medicines, School of Pharmaceutical Sciences, São Paulo State University, Araraquara, São Paulo, Brazil

  • Hérida R. Salgado,

    Roles Funding acquisition, Supervision, Writing – review & editing

    Affiliation Department of Drugs and Medicines, School of Pharmaceutical Sciences, São Paulo State University, Araraquara, São Paulo, Brazil

  • Hongfei Pi,

    Roles Data curation, Formal analysis, Investigation, Methodology

    Affiliation Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

  • Geoffrey W. Coombs,

    Roles Formal analysis, Resources, Writing – review & editing

    Affiliations Department of Microbiology, Path West Laboratory Medicine-WA, Fiona Stanley Hospital, Murdoch, Western Australia, Australia, School of Veterinary and Life Sciences, Murdoch University, Murdoch, Western Australia, Australia

  • Dean L. Shinabarger,

    Roles Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Resources, Supervision, Writing – review & editing

    Affiliation Micromyx LLC, Kalamazoo, Michighan, United States of America

  • John D. Turnidge,

    Roles Formal analysis, Validation, Writing – review & editing

    Affiliations Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia, Department of Molecular and Cellular Biology, School of Biological Sciences, The University of Adelaide, Adelaide, South Australia, Australia

  • James C. Paton ,

    Roles Conceptualization, Formal analysis, Funding acquisition, Resources, Supervision, Writing – review & editing

    ‡ These authors also contributed equally to this work.

    Affiliation Research Centre for Infectious Diseases, Department of Molecular and Cellular Biology, School of Biological Sciences, The University of Adelaide, Adelaide, South Australia, Australia

  • Adam McCluskey ,

    Roles Conceptualization, Formal analysis, Funding acquisition, Project administration, Resources, Software, Supervision, Writing – review & editing

    ‡ These authors also contributed equally to this work.

    Affiliation Chemistry, School of Environmental & Life Sciences, The University of Newcastle, Callaghan, New South Wales, Australia

  •  [ ... ],
  • Darren J. Trott

    Roles Conceptualization, Formal analysis, Funding acquisition, Project administration, Resources, Supervision, Writing – review & editing

    david.ogunniyi@adelaide.edu.au (ADO); darren.trott@adelaide.edu.au (DJT)

    ‡ These authors also contributed equally to this work.

    Affiliation Australian Centre for Antimicrobial Resistance Ecology, School of Animal and Veterinary Sciences, The University of Adelaide, Roseworthy, South Australia, Australia

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Evaluation of robenidine analog NCL195 as a novel broad-spectrum antibacterial agent

  • Abiodun D. Ogunniyi, 
  • Manouchehr Khazandi, 
  • Andrew J. Stevens, 
  • Sarah K. Sims, 
  • Stephen W. Page, 
  • Sanjay Garg, 
  • Henrietta Venter, 
  • Andrew Powell, 
  • Karen White, 
  • Kiro R. Petrovski
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