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Open Access
Peer-reviewed
Research Article
New 2-Ethylthio-4-methylaminoquinazoline derivatives inhibiting two subunits of cytochrome bc1 in Mycobacterium tuberculosis
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Andréanne Lupien ,
Contributed equally to this work with: Andréanne Lupien, Caroline Shi-Yan Foo
Roles Conceptualization, Formal analysis, Investigation, Methodology, Project administration, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
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Caroline Shi-Yan Foo ,
Contributed equally to this work with: Andréanne Lupien, Caroline Shi-Yan Foo
Roles Investigation, Methodology, Validation, Writing – original draft, Writing – review & editing
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
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Svetlana Savina,
Roles Investigation, Methodology
Affiliation Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation
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Anthony Vocat,
Roles Investigation, Methodology, Validation
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
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Jérémie Piton,
Roles Data curation, Methodology, Software
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
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Natalia Monakhova,
Roles Investigation, Methodology
Affiliation Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation
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Andrej Benjak,
Roles Data curation, Formal analysis, Software
Affiliation Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland
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Dirk A. Lamprecht,
Roles Investigation, Methodology, Writing – review & editing
Current address: Janssen Pharmaceutica, Beerse, Belgium.
Affiliation Africa Health Research Institute, Durban, South Africa
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Adrie J. C. Steyn,
Roles Supervision
Affiliations Africa Health Research Institute, Durban, South Africa, Department of Microbiology, University of Alabama at Birmingham, Birmingham, Alabama, United States of America
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Kevin Pethe,
Roles Validation
Affiliation Lee Kong Chian School of Medicine and School of Biological Sciences, Nanyang Technological University, Singapore
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Vadim A. Makarov ,
Roles Conceptualization, Investigation, Methodology, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: makarov@inbi.ras.ru (VAM); stewart.cole@pasteur.fr (STC)
Affiliation Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation
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Stewart T. Cole
Roles Conceptualization, Funding acquisition, Project administration, Resources, Supervision, Writing – review & editing
* E-mail: makarov@inbi.ras.ru (VAM); stewart.cole@pasteur.fr (STC)
Affiliations Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland, Institut Pasteur, rue du Docteur Roux, France
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New 2-Ethylthio-4-methylaminoquinazoline derivatives inhibiting two subunits of cytochrome bc1 in Mycobacterium tuberculosis
- Andréanne Lupien,
- Caroline Shi-Yan Foo,
- Svetlana Savina,
- Anthony Vocat,
- Jérémie Piton,
- Natalia Monakhova,
- Andrej Benjak,
- Dirk A. Lamprecht,
- Adrie J. C. Steyn,
- Kevin Pethe
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- Published: January 23, 2020
- https://doi.org/10.1371/journal.ppat.1008270