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Open Access
Peer-reviewed
Research Article
The trypanocidal benzoxaborole AN7973 inhibits trypanosome mRNA processing
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Daniela Begolo,
Roles Conceptualization, Formal analysis, Investigation, Methodology, Visualization, Writing – original draft, Writing – review & editing
Affiliation Center for Molecular Biology of Heidelberg University (ZMBH), DKFZ-ZMBH Alliance, Im Neuenheimer Feld 282, Heidelberg, Germany
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Isabel M. Vincent,
Roles Investigation, Writing – original draft, Writing – review & editing
Affiliation Wellcome Centre for Molecular Parasitology, Institute of Infection, Immunity and Inflammation, College of Medical, Veterinary and Life Sciences, 120 University Place, University of Glasgow, Glasgow, United Kingdom
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Federica Giordani,
Roles Investigation, Writing – original draft, Writing – review & editing
Affiliation Wellcome Centre for Molecular Parasitology, Institute of Infection, Immunity and Inflammation, College of Medical, Veterinary and Life Sciences, 120 University Place, University of Glasgow, Glasgow, United Kingdom
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Ina Pöhner,
Roles Formal analysis, Investigation, Methodology, Visualization, Writing – original draft, Writing – review & editing
Affiliation Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies (HITS), Schloß-Wolfsbrunnenweg 35, Heidelberg, Germany
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Michael J. Witty,
Roles Conceptualization, Funding acquisition, Methodology, Project administration, Supervision, Writing – review & editing
Affiliation Global Alliance for Livestock and Veterinary Medicine, Doherty Building, Pentlands Science Park, Penicuik, Edinburgh, United Kingdom
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Timothy G. Rowan,
Roles Conceptualization, Funding acquisition, Methodology, Project administration, Writing – original draft, Writing – review & editing
Affiliation Global Alliance for Livestock and Veterinary Medicine, Doherty Building, Pentlands Science Park, Penicuik, Edinburgh, United Kingdom
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Zakaria Bengaly,
Roles Investigation
Affiliation Centre International de Recherche–Développement sur l’Elevage en zone Subhumide (CIRDES), Bobo-Dioulasso 01, Burkina Faso
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Kirsten Gillingwater,
Roles Investigation, Methodology, Writing – original draft, Writing – review & editing
Affiliations Swiss Tropical and Public Health Institute, Socinstrasse 57, Basel, Switzerland, University of Basel, Petersplatz 1, Basel, Switzerland
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Yvonne Freund,
Roles Formal analysis, Resources, Writing – review & editing
Current address: Los Altos, CA, United States of America
Affiliation Anacor Pharmaceuticals, Inc., Palo Alto, CA, United States of America
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Rebecca C. Wade,
Roles Formal analysis, Investigation, Methodology, Supervision, Visualization, Writing – original draft, Writing – review & editing
Affiliations Center for Molecular Biology of Heidelberg University (ZMBH), DKFZ-ZMBH Alliance, Im Neuenheimer Feld 282, Heidelberg, Germany, Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies (HITS), Schloß-Wolfsbrunnenweg 35, Heidelberg, Germany, Interdisciplinary Center for Scientific Computing (IWR), Heidelberg University, Im Neuenheimer Feld 205, Heidelberg, Germany
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Michael P. Barrett,
Roles Conceptualization, Formal analysis, Funding acquisition, Methodology, Project administration, Supervision, Visualization, Writing – original draft, Writing – review & editing
Affiliations Wellcome Centre for Molecular Parasitology, Institute of Infection, Immunity and Inflammation, College of Medical, Veterinary and Life Sciences, 120 University Place, University of Glasgow, Glasgow, United Kingdom, Glasgow Polyomics, University of Glasgow, Glasgow, United Kingdom
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Christine Clayton
Roles Conceptualization, Formal analysis, Funding acquisition, Methodology, Project administration, Supervision, Visualization, Writing – original draft, Writing – review & editing
* E-mail: cclayton@zmbh.uni-heidelberg.de
Affiliation Center for Molecular Biology of Heidelberg University (ZMBH), DKFZ-ZMBH Alliance, Im Neuenheimer Feld 282, Heidelberg, Germany
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The trypanocidal benzoxaborole AN7973 inhibits trypanosome mRNA processing
- Daniela Begolo,
- Isabel M. Vincent,
- Federica Giordani,
- Ina Pöhner,
- Michael J. Witty,
- Timothy G. Rowan,
- Zakaria Bengaly,
- Kirsten Gillingwater,
- Yvonne Freund,
- Rebecca C. Wade
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- Published: September 25, 2018
- https://doi.org/10.1371/journal.ppat.1007315
- See the preprint