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Open Access
Peer-reviewed
Research Article
Two key cathepsins, TgCPB and TgCPL, are targeted by the vinyl sulfone inhibitor K11777 in in vitro and in vivo models of toxoplasmosis
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Juan D. Chaparro,
Roles Conceptualization, Formal analysis, Investigation, Methodology, Writing – original draft, Writing – review & editing
Current address: Nationwide Children’s Hospital, 700 Children’s Dr., Columbus, Ohio, United States of America
Affiliation Department of Pediatrics, Division of Infectious Diseases, Rady Children's Hospital, University of California, San Diego, School of Medicine, La Jolla, California, United States of America
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Timmy Cheng,
Roles Conceptualization, Data curation, Investigation, Methodology, Writing – original draft, Writing – review & editing
Current address: Department of Medicine, Division of Pulmonary Medicine and Critical Care, University of California Irvine, Irvine, California, United States of America
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Uyen Phuong Tran,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Writing – original draft
Current address: Department of Pathology, University of California Irvine School of Medicine, Irvine, California, United States of America
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Rosa M. Andrade,
Roles Data curation, Formal analysis, Investigation, Methodology, Writing – original draft, Writing – review & editing
Affiliation Department of Medicine, Division of Infectious Diseases, University of California, Irvine School of Medicine, Irvine, California, United States of America
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Sara B. T. Brenner,
Roles Data curation, Formal analysis, Investigation, Methodology, Writing – original draft, Writing – review & editing
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Grace Hwang,
Roles Investigation, Methodology, Writing – original draft, Writing – review & editing
Current address: Illumina, Inc., San Diego, California, United States of America
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Shara Cohn,
Roles Data curation, Investigation, Methodology, Writing – review & editing
Current address: Department of Anesthesiology, Stanford University School of Medicine, Stanford, California, United States of America
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Ken Hirata,
Roles Conceptualization, Data curation, Formal analysis, Methodology, Project administration, Writing – original draft, Writing – review & editing
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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James H. McKerrow,
Roles Conceptualization, Funding acquisition, Resources, Writing – original draft, Writing – review & editing
Affiliation Department of Pharmacy, Skaggs School of Pharmacy and Pharmaceutical Science, University of California, San Diego, La Jolla, California, United States of America
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Sharon L. Reed
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing
* E-mail: slreed@ucsd.edu
Affiliation Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America
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Two key cathepsins, TgCPB and TgCPL, are targeted by the vinyl sulfone inhibitor K11777 in in vitro and in vivo models of toxoplasmosis
- Juan D. Chaparro,
- Timmy Cheng,
- Uyen Phuong Tran,
- Rosa M. Andrade,
- Sara B. T. Brenner,
- Grace Hwang,
- Shara Cohn,
- Ken Hirata,
- James H. McKerrow,
- Sharon L. Reed
- Published: March 22, 2018
- https://doi.org/10.1371/journal.pone.0193982