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Open Access
Peer-reviewed
Research Article
Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice
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Stefan Just ,
Contributed equally to this work with: Stefan Just, Bertrand L. Chenard
Roles Conceptualization, Data curation, Formal analysis, Investigation, Project administration, Supervision, Writing – original draft, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Bertrand L. Chenard ,
Contributed equally to this work with: Stefan Just, Bertrand L. Chenard
Roles Conceptualization, Data curation, Project administration, Supervision, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Angelo Ceci,
Roles Conceptualization, Formal analysis, Investigation, Project administration, Supervision, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Timothy Strassmaier,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Project administration, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Jayhong A. Chong,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Methodology, Project administration, Writing – original draft, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Nathaniel T. Blair,
Roles Data curation, Formal analysis, Investigation, Methodology, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Randall J. Gallaschun,
Roles Conceptualization, Investigation, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Donato del Camino,
Roles Conceptualization, Formal analysis, Investigation, Methodology, Project administration, Supervision, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Susan Cantin,
Roles Data curation, Formal analysis, Supervision
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Marc D’Amours,
Roles Investigation, Methodology
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Christian Eickmeier,
Roles Conceptualization, Project administration, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Christopher M. Fanger,
Roles Data curation, Project administration, Supervision
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Carsten Hecker,
Roles Formal analysis, Investigation, Methodology
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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David P. Hessler,
Roles Investigation, Project administration, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Bastian Hengerer,
Roles Conceptualization, Project administration, Supervision
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Katja S. Kroker,
Roles Formal analysis, Investigation, Project administration, Supervision, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Sam Malekiani,
Roles Project administration, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Robert Mihalek,
Roles Formal analysis, Investigation, Methodology
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Joseph McLaughlin,
Roles Formal analysis, Investigation, Methodology
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Georg Rast,
Roles Data curation, Investigation, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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JoAnn Witek,
Roles Investigation, Methodology, Supervision, Writing – review & editing
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Achim Sauer,
Roles Conceptualization, Data curation, Formal analysis, Methodology, Project administration, Resources, Supervision, Writing – original draft, Writing – review & editing
Affiliation Boehringer Ingelheim Pharma GmbH & Co. KG, Biberach an der Riss, Germany
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Christopher R. Pryce,
Roles Conceptualization, Data curation, Formal analysis, Methodology, Supervision, Writing – original draft, Writing – review & editing
Affiliation Preclinical Laboratory for Translational Research into Affective Disorders, Department of Psychiatry, Psychotherapy & Psychosomatics, Psychiatric Hospital, University of Zurich, Zurich, Switzerland
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Magdalene M. Moran
Roles Conceptualization, Data curation, Project administration, Supervision, Writing – original draft, Writing – review & editing
* E-mail: mmoran@hydrabiosciences.com
Affiliation Hydra Biosciences, Cambridge, Massachusetts, United States of America
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Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice
- Stefan Just,
- Bertrand L. Chenard,
- Angelo Ceci,
- Timothy Strassmaier,
- Jayhong A. Chong,
- Nathaniel T. Blair,
- Randall J. Gallaschun,
- Donato del Camino,
- Susan Cantin,
- Marc D’Amours
- Published: January 31, 2018
- https://doi.org/10.1371/journal.pone.0191225