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Open Access
Peer-reviewed
Research Article
The Open Form Inducer Approach for Structure-Based Drug Design
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Daniel Ken Inaoka ,
* E-mail: danielken@nagasaki-u.ac.jp
Affiliations School of Tropical Medicine and Global Health, Nagasaki University, Nagasaki, Japan, Department of Biomedical Chemistry, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan
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Maiko Iida,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Toshiyuki Tabuchi,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Teruki Honma,
Affiliation Systems and Structural Biology Center, RIKEN, Tsurumi, Yokohama, Japan
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Nayoung Lee,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Satoshi Hashimoto,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Shigeru Matsuoka,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Takefumi Kuranaga,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Kazuhito Sato,
Affiliation Systems and Structural Biology Center, RIKEN, Tsurumi, Yokohama, Japan
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Tomoo Shiba,
Affiliation Department of Applied Biology, Graduate School of Science and Technology, Kyoto Institute of Technology, Kyoto, Japan
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Kimitoshi Sakamoto,
Affiliation Department of Biochemistry and Molecular Biology, Faculty of Agriculture and Life Science, Hirosaki University, Aomori, Japan
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Emmanuel Oluwadare Balogun,
Affiliation Department of Biomedical Chemistry, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan
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Shigeo Suzuki,
Affiliation Department of Biomedical Chemistry, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan
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Takeshi Nara,
Affiliation Department of Molecular and Cellular Parasitology, Juntendo University School of Medicine, Tokyo, Japan
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Josmar Rodrigues da Rocha,
Affiliation Institute of Chemistry of São Carlos, University of São Paulo, São Paulo, Brazil
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Carlos Alberto Montanari,
Affiliation Institute of Chemistry of São Carlos, University of São Paulo, São Paulo, Brazil
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Akiko Tanaka,
Affiliation Systems and Structural Biology Center, RIKEN, Tsurumi, Yokohama, Japan
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Masayuki Inoue,
Affiliation Department of Integrated Analytical Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo, Japan
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Kiyoshi Kita,
Affiliations School of Tropical Medicine and Global Health, Nagasaki University, Nagasaki, Japan, Department of Biomedical Chemistry, Graduate School of Medicine, The University of Tokyo, Tokyo, Japan
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Shigeharu Harada
Affiliation Department of Applied Biology, Graduate School of Science and Technology, Kyoto Institute of Technology, Kyoto, Japan
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The Open Form Inducer Approach for Structure-Based Drug Design
- Daniel Ken Inaoka,
- Maiko Iida,
- Toshiyuki Tabuchi,
- Teruki Honma,
- Nayoung Lee,
- Satoshi Hashimoto,
- Shigeru Matsuoka,
- Takefumi Kuranaga,
- Kazuhito Sato,
- Tomoo Shiba
- Published: November 28, 2016
- https://doi.org/10.1371/journal.pone.0167078