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Open Access
Peer-reviewed
Research Article
AMPK Activation through Mitochondrial Regulation Results in Increased Substrate Oxidation and Improved Metabolic Parameters in Models of Diabetes
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Yonchu Jenkins ,
Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Tian-Qiang Sun ,
Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Vadim Markovtsov ,
Contributed equally to this work with: Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Marc Foretz,
Affiliations Inserm, U1016, Institut Cochin, Paris, France, CNRS, UMR8104, Paris, France, Université Paris Descartes, Sorbonne Paris cité, Paris, France
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Wei Li,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Henry Nguyen,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Yingwu Li,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Alison Pan,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Gerald Uy,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Lisa Gross,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Kristen Baltgalvis,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Stephanie L. Yung,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Tarikere Gururaja,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Taisei Kinoshita,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Alexander Owyang,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Ira J. Smith,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Kelly McCaughey,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Kathy White,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Guillermo Godinez,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Raniel Alcantara,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Carmen Choy,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Hong Ren,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Rachel Basile,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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David J. Sweeny,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Xiang Xu,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Sarkiz D. Issakani,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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David C. Carroll,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Dane A. Goff,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Simon J. Shaw,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Rajinder Singh,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Laszlo G. Boros,
Affiliations SiDMAP, LLC, Los Angeles, California, United States of America, Department of Pediatrics, Los Angeles Biomedical Research Institute (LABIOMED) at the Harbor-UCLA Medical Center, Torrance, California, United States of America
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Marc-André Laplante,
Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
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Bruno Marcotte,
Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
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Rita Kohen,
Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
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Benoit Viollet,
Affiliations Inserm, U1016, Institut Cochin, Paris, France, CNRS, UMR8104, Paris, France, Université Paris Descartes, Sorbonne Paris cité, Paris, France
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André Marette,
Affiliation Department of Medicine, Faculty of Medicine, Cardiology Axis of the Institut Universitaire de Cardiologie et de Pneumologie de Québec (Hôpital Laval), Québec, Québec, Canada
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Donald G. Payan,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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Todd M. Kinsella,
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
⨯ - [ ... ],
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Yasumichi Hitoshi
* E-mail: yhitoshi@rigel.com
Affiliation Rigel Pharmaceuticals, Inc., South San Francisco, California, United States of America
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AMPK Activation through Mitochondrial Regulation Results in Increased Substrate Oxidation and Improved Metabolic Parameters in Models of Diabetes
- Yonchu Jenkins,
- Tian-Qiang Sun,
- Vadim Markovtsov,
- Marc Foretz,
- Wei Li,
- Henry Nguyen,
- Yingwu Li,
- Alison Pan,
- Gerald Uy,
- Lisa Gross
- Published: December 5, 2013
- https://doi.org/10.1371/journal.pone.0081870