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Open Access
Peer-reviewed
Research Article
Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors
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Thomas W. Miller ,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Methodology, Project administration, Resources, Supervision, Validation, Visualization, Writing – original draft, Writing – review & editing
* E-mail: thomas.miller@pstherx.com
Affiliations Paradigm Shift Therapeutics LLC, Rockville, Maryland, United States of America, Laboratory of Pathology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland, United States of America
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Joshua D. Amason,
Roles Data curation, Investigation, Methodology, Writing – review & editing
Current address: Department of Ophthalmology, Duke University School of Medicine, Durham, North Carolina, United States of America
Affiliations Paradigm Shift Therapeutics LLC, Rockville, Maryland, United States of America, Laboratory of Pathology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland, United States of America
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Elsa D. Garcin,
Roles Conceptualization, Investigation, Methodology, Resources, Visualization, Writing – review & editing
Affiliation Department of Chemistry and Biochemistry, University of Maryland Baltimore County, Catonsville, Maryland, United States of America
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Laurence Lamy,
Roles Investigation, Writing – review & editing
Affiliation Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Patricia K. Dranchak,
Roles Conceptualization, Data curation, Formal analysis, Software, Visualization, Writing – review & editing
Affiliation Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Ryan Macarthur,
Roles Data curation, Formal analysis, Methodology, Software, Visualization, Writing – review & editing
Affiliation Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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John Braisted,
Roles Data curation, Formal analysis, Software, Visualization
Affiliation Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Jeffrey S. Rubin,
Roles Conceptualization, Funding acquisition, Methodology, Writing – original draft, Writing – review & editing
Affiliation Paradigm Shift Therapeutics LLC, Rockville, Maryland, United States of America
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Teresa L. Burgess,
Roles Conceptualization, Funding acquisition, Methodology, Project administration, Writing – original draft, Writing – review & editing
Affiliation Paradigm Shift Therapeutics LLC, Rockville, Maryland, United States of America
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Catherine L. Farrell,
Roles Conceptualization, Funding acquisition, Methodology, Project administration, Resources, Writing – review & editing
Affiliation Paradigm Shift Therapeutics LLC, Rockville, Maryland, United States of America
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David D. Roberts,
Roles Conceptualization, Methodology, Resources, Writing – review & editing
Affiliation Laboratory of Pathology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland, United States of America
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James Inglese
Roles Conceptualization, Formal analysis, Methodology, Project administration, Resources, Supervision, Visualization, Writing – original draft, Writing – review & editing
Affiliation Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors
- Thomas W. Miller,
- Joshua D. Amason,
- Elsa D. Garcin,
- Laurence Lamy,
- Patricia K. Dranchak,
- Ryan Macarthur,
- John Braisted,
- Jeffrey S. Rubin,
- Teresa L. Burgess,
- Catherine L. Farrell
- Published: July 5, 2019
- https://doi.org/10.1371/journal.pone.0218897