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Open Access
Peer-reviewed
Research Article
Specific blockade of Rictor-mTOR association inhibits mTORC2 activity and is cytotoxic in glioblastoma
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Angelica Benavides-Serrato ,
Contributed equally to this work with: Angelica Benavides-Serrato, Jihye Lee
Affiliations Department of Medicine, David Geffen School of Medicine, University of California-Los Angeles, Los Angeles, California, United States of America, Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America
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Jihye Lee ,
Contributed equally to this work with: Angelica Benavides-Serrato, Jihye Lee
Current address: Neuroscience Research Institute, Gachon University, 24, Namdong-daero 774 beon-gil, Namdong-gu, Incheon, South Korea
Affiliation Department of Chemistry and Biochemistry, University of California-Los Angeles, Los Angeles, California, United States of America
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Brent Holmes,
Affiliations Department of Medicine, David Geffen School of Medicine, University of California-Los Angeles, Los Angeles, California, United States of America, Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America
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Kenna A. Landon,
Affiliation Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America
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Tariq Bashir,
Affiliation Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America
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Michael E. Jung,
Affiliations Department of Chemistry and Biochemistry, University of California-Los Angeles, Los Angeles, California, United States of America, Jonnson Comprehensive Cancer Center, University of California-Los Angeles, Los Angeles, California, United States of America, Molecular Biology Institute, University of California-Los Angeles, Los Angeles, California, United States of America
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Alan Lichtenstein,
Affiliations Department of Medicine, David Geffen School of Medicine, University of California-Los Angeles, Los Angeles, California, United States of America, Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America, Jonnson Comprehensive Cancer Center, University of California-Los Angeles, Los Angeles, California, United States of America
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Joseph Gera
* E-mail: jgera@mednet.ucla.edu
Affiliations Department of Medicine, David Geffen School of Medicine, University of California-Los Angeles, Los Angeles, California, United States of America, Department of Research & Development, Greater Los Angeles Veterans Affairs Healthcare System, Los Angeles, California, United States of America, Jonnson Comprehensive Cancer Center, University of California-Los Angeles, Los Angeles, California, United States of America, Molecular Biology Institute, University of California-Los Angeles, Los Angeles, California, United States of America
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Specific blockade of Rictor-mTOR association inhibits mTORC2 activity and is cytotoxic in glioblastoma
- Angelica Benavides-Serrato,
- Jihye Lee,
- Brent Holmes,
- Kenna A. Landon,
- Tariq Bashir,
- Michael E. Jung,
- Alan Lichtenstein,
- Joseph Gera
- Published: April 28, 2017
- https://doi.org/10.1371/journal.pone.0176599