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Open Access
Peer-reviewed
Research Article
A Homogeneous, High-Throughput Assay for Phosphatidylinositol 5-Phosphate 4-Kinase with a Novel, Rapid Substrate Preparation
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Mindy I. Davis ,
Contributed equally to this work with: Mindy I. Davis, Atsuo T. Sasaki
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Atsuo T. Sasaki ,
Contributed equally to this work with: Mindy I. Davis, Atsuo T. Sasaki
Affiliations Beth Israel Deaconess Medical Center, Department of Medicine, Division of Signal Transduction; Department of Systems Biology, Harvard Medical School, Boston, Massachusetts, United States of America, Division of Hematology and Oncology, Department of Internal Medicine, Neuroscience Institute: Brain Tumor Center, University of Cincinnati, College of Medicine, Cincinnati, Ohio, United States of America
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Min Shen,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Brooke M. Emerling,
Affiliation Beth Israel Deaconess Medical Center, Department of Medicine, Division of Signal Transduction; Department of Systems Biology, Harvard Medical School, Boston, Massachusetts, United States of America
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Natasha Thorne,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Sam Michael,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Rajan Pragani,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Matthew Boxer,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Kazutaka Sumita,
Affiliation Division of Hematology and Oncology, Department of Internal Medicine, Neuroscience Institute: Brain Tumor Center, University of Cincinnati, College of Medicine, Cincinnati, Ohio, United States of America
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Koh Takeuchi,
Affiliation Biomedicinal Information Research Center, National Institute of Advanced Industrial Science and Technology, Koto, Tokyo, Japan
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Douglas S. Auld,
Affiliations National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America, Center for Proteomic Chemistry, Novartis Institutes for Biomedical Research, Cambridge, Massachusetts, United States of America
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Zhuyin Li,
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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Lewis C. Cantley,
Affiliation Beth Israel Deaconess Medical Center, Department of Medicine, Division of Signal Transduction; Department of Systems Biology, Harvard Medical School, Boston, Massachusetts, United States of America
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Anton Simeonov
* E-mail: asimeono@mail.nih.gov
Affiliation National Institutes of Health Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, United States of America
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A Homogeneous, High-Throughput Assay for Phosphatidylinositol 5-Phosphate 4-Kinase with a Novel, Rapid Substrate Preparation
- Mindy I. Davis,
- Atsuo T. Sasaki,
- Min Shen,
- Brooke M. Emerling,
- Natasha Thorne,
- Sam Michael,
- Rajan Pragani,
- Matthew Boxer,
- Kazutaka Sumita,
- Koh Takeuchi

- Published: January 10, 2013
- https://doi.org/10.1371/journal.pone.0054127