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Open Access
Peer-reviewed
Research Article
Epidermal Growth Factor Receptor Activation in Glioblastoma through Novel Missense Mutations in the Extracellular Domain
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Jeffrey C Lee,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Department of Pathology, Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Igor Vivanco,
Affiliation Department of Molecular & Medical Pharmacology, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Rameen Beroukhim,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America , Department of Medicine, Harvard Medical School, Boston, Massachusetts, United States of America
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Julie H. Y Huang,
Affiliation Department of Human Genetics, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Whei L Feng,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Ralph M DeBiasi,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Koji Yoshimoto,
Affiliation Department of Pathology and Laboratory Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Jennifer C King,
Affiliation Department of Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Phioanh Nghiemphu,
Affiliation Department of Neurology, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Yuki Yuza,
Affiliation Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America
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Qing Xu,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Department of Medicine, Harvard Medical School, Boston, Massachusetts, United States of America
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Heidi Greulich,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America , Department of Medicine, Harvard Medical School, Boston, Massachusetts, United States of America
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Roman K Thomas,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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J. Guillermo Paez,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America , Department of Medicine, Harvard Medical School, Boston, Massachusetts, United States of America
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Timothy C Peck,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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David J Linhart,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Karen A Glatt,
Affiliation Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America
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Gad Getz,
Affiliation Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Robert Onofrio,
Affiliation Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Liuda Ziaugra,
Affiliation Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Ross L Levine,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Department of Medicine, Brigham and Women's Hospital, Boston, Massachusetts, United States of America
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Stacey Gabriel,
Affiliation Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Tomohiro Kawaguchi,
Affiliation Department of Neurosurgery, University of California San Francisco, San Francisco, California, United States of America
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Keith O'Neill,
Affiliation Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Haumith Khan,
Affiliation Department of Neurosurgery, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Linda M Liau,
Affiliation Department of Neurosurgery, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Stanley F Nelson,
Affiliation Department of Human Genetics, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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P. Nagesh Rao,
Affiliation Department of Pathology and Laboratory Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Paul Mischel,
Affiliation Department of Pathology and Laboratory Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Russell O Pieper,
Affiliation Department of Neurosurgery, University of California San Francisco, San Francisco, California, United States of America
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Tim Cloughesy,
Affiliation Department of Neurology, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Daniel J Leahy,
Affiliations Department of Biophysics and Biophysical Chemistry, The Johns Hopkins University School of Medicine, Baltimore, Maryland, United States of America , Howard Hughes Medical Institute, The Johns Hopkins University School of Medicine, Baltimore, Maryland, United States of America
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William R Sellers,
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America , Department of Medicine, Harvard Medical School, Boston, Massachusetts, United States of America
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Charles L Sawyers,
Affiliations Department of Molecular & Medical Pharmacology, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America , Department of Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America , Howard Hughes Medical Institute, University of California Los Angeles, Los Angeles, California, United States of America
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Matthew Meyerson ,
*To whom correspondence should be addressed. E-mail: matthew_meyerson@dfci.harvard.edu (MM); imellinghoff@mednet.ucla.edu (IKM)
Affiliations Department of Medical Oncology and Center for Cancer Genome Discovery, Dana-Farber Cancer Institute Harvard Medical School, Boston, Massachusetts, United States of America , Department of Pathology, Harvard Medical School, Boston, Massachusetts, United States of America , Broad Institute of Harvard and Massachusetts Institute of Technology, Cambridge, Massachusetts, United States of America
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Ingo K Mellinghoff
*To whom correspondence should be addressed. E-mail: matthew_meyerson@dfci.harvard.edu (MM); imellinghoff@mednet.ucla.edu (IKM)
Affiliations Department of Molecular & Medical Pharmacology, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America , Department of Medicine, David Geffen School of Medicine, University of California Los Angeles, Los Angeles, California, United States of America
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Epidermal Growth Factor Receptor Activation in Glioblastoma through Novel Missense Mutations in the Extracellular Domain
- Jeffrey C Lee,
- Igor Vivanco,
- Rameen Beroukhim,
- Julie H. Y Huang,
- Whei L Feng,
- Ralph M DeBiasi,
- Koji Yoshimoto,
- Jennifer C King,
- Phioanh Nghiemphu,
- Yuki Yuza
- Published: December 19, 2006
- https://doi.org/10.1371/journal.pmed.0030485