-
Loading metrics
Open Access
Peer-reviewed
Research Article
Rational design of highly potent broad-spectrum enterovirus inhibitors targeting the nonstructural protein 2C
-
Lisa Bauer,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Roberto Manganaro,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Writing – original draft, Writing – review & editing
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Birgit Zonsics,
Roles Conceptualization, Data curation, Formal analysis, Investigation, Writing – original draft, Writing – review & editing
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Daniel L. Hurdiss,
Roles Conceptualization, Data curation, Formal analysis, Funding acquisition, Investigation, Validation, Visualization, Writing – original draft, Writing – review & editing
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Marleen Zwaagstra,
Roles Data curation, Investigation
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Tim Donselaar,
Roles Data curation, Investigation
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Naemi G. E. Welter,
Roles Data curation, Formal analysis, Investigation
Affiliation Neurotoxicology Research Group, Toxicology Division, Institute for Risk Assessment Sciences (IRAS), Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Regina G. D. M. van Kleef,
Roles Data curation, Formal analysis, Investigation
Affiliation Neurotoxicology Research Group, Toxicology Division, Institute for Risk Assessment Sciences (IRAS), Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Moira Lorenzo Lopez,
Roles Data curation, Investigation
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Federica Bevilacqua,
Roles Data curation, Investigation
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Thamidur Raman,
Roles Data curation, Investigation
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Salvatore Ferla,
Roles Conceptualization, Data curation, Investigation, Writing – original draft, Writing – review & editing
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ -
Marcella Bassetto,
Roles Data curation, Investigation
Affiliation Department of Chemistry, Swansea University, Swansea, United Kingdom
⨯ -
Johan Neyts,
Roles Conceptualization, Writing – review & editing
Affiliation Department of Microbiology, Immunology and Transplantation, Rega Institute for Medical Research, KU Leuven, Leuven, Belgium
⨯ -
Jeroen R. P. M. Strating,
Roles Conceptualization, Funding acquisition, Supervision
Current address: Viroclinics, Rotterdam, The Netherlands
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Remco H. S. Westerink,
Roles Conceptualization, Data curation, Formal analysis, Methodology, Supervision, Writing – original draft, Writing – review & editing
Affiliation Neurotoxicology Research Group, Toxicology Division, Institute for Risk Assessment Sciences (IRAS), Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ -
Andrea Brancale,
Roles Conceptualization, Funding acquisition, Investigation, Methodology, Supervision, Validation, Writing – original draft, Writing – review & editing
Affiliation Medicinal Chemistry, School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Cardiff, United Kingdom
⨯ - [ ... ],
-
Frank J. M. van Kuppeveld
Roles Conceptualization, Funding acquisition, Investigation, Methodology, Supervision, Validation, Writing – original draft, Writing – review & editing
* E-mail: f.j.m.vankuppeveld@uu.nl
Affiliation Virology Section, Infectious Disease and Immunology Division, Department of Biomolecular Health Sciences, Faculty of Veterinary Medicine, Utrecht University, Utrecht, The Netherlands
⨯ - [ view all ]
- [ view less ]
Rational design of highly potent broad-spectrum enterovirus inhibitors targeting the nonstructural protein 2C
- Lisa Bauer,
- Roberto Manganaro,
- Birgit Zonsics,
- Daniel L. Hurdiss,
- Marleen Zwaagstra,
- Tim Donselaar,
- Naemi G. E. Welter,
- Regina G. D. M. van Kleef,
- Moira Lorenzo Lopez,
- Federica Bevilacqua
-
- Published: November 6, 2020
- https://doi.org/10.1371/journal.pbio.3000904